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1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-2-one
2-cyclopropyl-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}pyrimidine-5-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propylsulfanyl)ethan-1-one
(4aR,7aS)-1-(2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]benzamide
N-(2-methoxyethyl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(3-phenylprop-2-yn-1-yl)acetamide
N-(4-methoxy-2-methylphenyl)-3-[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]propanamide
(1S,6R)-9-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
6-{[5-(furan-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
1-{1-oxo-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-2-yl}pyrrolidin-2-one
3,5-dimethyl-2-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
3-{ethyl[(2-fluorophenyl)methyl]amino}propane-1,2-diol
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
6-[(2-hydroxy-6-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-cyclopropyl-4-fluoro-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]benzamide
1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}-4-methylpiperidine
N-methyl-1-(naphthalen-1-ylmethyl)-N-(oxolan-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
4-[(3-chlorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
(3R,4R)-N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carboxamide
4-[3-(furan-2-yl)-3-phenylpropanoyl]-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(1S,5R)-6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}benzamide
(3S,4R)-N,N-dimethyl-1-[(5-methylthiophen-2-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-amine
3-chloro-N-cyclopentyl-4-({1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
1-({4-[(5-cyanopyridin-2-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-4-oxo-4H-chromene-2-carboxamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperidine-4-carboxylic acid
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(4-phenylbutan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-benzoyl-1-benzofuran-3-yl)methyl]-4-ethylpiperazine-2,3-dione
5-(1,3-benzothiazol-2-ylmethyl)-1-(cyclopropylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3-methylphenyl)-4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-(1H-imidazol-2-ylmethyl)-3-(4-methoxyphenyl)-3-phenylpropanamide
2-[2-methyl-3-({2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-indol-1-yl]acetamide
4-[6-(propan-2-yl)pyridazin-3-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
3-{5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-{1-[(2-ethoxyphenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
2-acetamido-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
(1S,5R)-3-(2-amino-6-methoxypyrimidin-4-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-{6-[4-(aminomethyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)-1H-pyrazole
N-cyclopropyl-3-({1-[(4-acetamidophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
9-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
(2S)-1-(1-methylpiperidin-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidine-2-carboxamide
2-ethyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide