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3-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-{[(1-hydroxybutan-2-yl)(thiophen-2-ylmethyl)amino]methyl}-6-methylphenol
{3-[(3-chlorophenyl)methyl]-1-(2,6-diaminopyrimidin-4-yl)piperidin-3-yl}methanol
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-4-(4-fluorophenyl)butane-1,4-dione
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-methyl-4-({5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methyl)piperazine
1-[(3-chlorophenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
6-tert-butyl-1-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)phenyl]ethan-1-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(3-fluoro-4-methoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
5-(1-{2-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-3-methyl-1,2,4-oxadiazole
1-[(3-methylphenyl)methyl]-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
4,6-dimethyl-2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyridine-3-carbonitrile
1-[(4-methyl-5-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
(4aR,7aS)-1-{2-[4-(hydroxymethyl)piperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[2-(2-fluorophenyl)ethyl]acetamide
2-(2,5-dimethylphenoxy)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]propanamide
2-[(3-methoxyphenyl)sulfanyl]-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
1-[4-benzyl-4-(hydroxymethyl)piperidine-1-carbonyl]-7-chloro-9H-fluoren-9-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-(2-phenylpropyl)-1H-1,3-benzodiazole-7-carboxamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-amino-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)-6-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridine-3-carbonitrile
2-(4-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
1,6-dimethyl-2-oxo-N-(2-phenylpropyl)-1,2-dihydropyridine-3-carboxamide
2,4-dimethyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)pyrimidine-5-carboxamide
1-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-2,3-dihydro-1H-indole
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(morpholin-2-yl)ethan-1-one
[(2S)-1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
3-chloro-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[2-(4H-1,2,4-triazol-4-yl)benzoyl]thiomorpholine
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(propan-2-ylsulfanyl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
6-{[4-(2-ethyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]methyl}quinoxaline
5-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(4-fluorophenyl)-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
2-[3-(2-chlorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-(dicyclopropylmethyl)-N-methylacetamide
1-cyclopentyl-N5-[(2-methoxyphenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,4-difluorophenyl)-5-[(5-fluoro-2-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[2-(dimethylamino)ethyl]-5-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine
7-methyl-2-(1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,3-benzothiazole-6-carboxamide
N-cyclopropyl-5-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1'-[(2-fluoro-4-methoxyphenyl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(1-benzylpiperidin-3-yl)methyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine