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(5S)-5-[({[2-(methylsulfanyl)pyrimidin-5-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
7-fluoro-4-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)quinazoline
N-(2-methoxyethyl)-4-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-2-carboxamide
1-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-ethylpiperidine-3-carboxylic acid
1-(oxolane-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]cyclopropane-1-carboxamide
N-cyclohexyl-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]propanamide
4-methyl-2-{[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5,6,7,8-tetrahydroquinazoline
2-ethyl-8-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]acetamide
1-[(2-ethylphenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
6-(1-benzothiophen-7-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-methyl-7-(4-methyl-1H-imidazole-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
6-fluoro-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(4-chloro-3-methylphenyl)-2-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
(2S)-2-[(2-oxo-6-phenyl-1,2-dihydropyridin-3-yl)formamido]-3-phenylpropanamide
(1R,5R)-3-(2-methoxy-5-methylbenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-(2-fluorophenyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-(morpholin-4-yl)-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propan-1-one
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
N-cyclobutyl-4-[(pyridin-2-ylmethyl)sulfamoyl]benzamide
(1R,5R)-3-[4-(1H-imidazol-1-yl)benzoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
(2R)-2-[5-(2-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
5-methyl-2-(2-phenylphenyl)pyrimidin-4-amine
N-[(3R,4S)-4-(propan-2-yl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]methanesulfonamide
(4aS,8aS)-N-cyclohexyl-4a-hydroxy-7-(pyridin-2-yl)-decahydro-2,7-naphthyridine-2-carboxamide
(3S,4R)-1-(7-chloro-1-methyl-1H-indole-2-carbonyl)-3-ethyl-4-methylpiperidin-4-ol
N-[(1-phenylcyclopentyl)methyl]-6-(quinolin-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
dimethyl({[4-methyl-5-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
3,4,7-trimethyl-N-[(1-methyl-5-oxopyrrolidin-2-yl)methyl]-1H-indole-2-carboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-ethyl-3-(1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanoyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-oxo-1-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxylic acid
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-(cyclopropylmethyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
3-{1-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-N,N-diethyl-1-(2-methanesulfonylacetyl)pyrrolidine-2-carboxamide
3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
1-benzoyl-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidin-4-amine
2-methyl-3-(1H-pyrazol-3-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine
3-[(2-fluorophenyl)formamido]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-(furan-2-ylmethyl)piperidine-4-carboxamide
4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one