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3-[5-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-(1-methyl-1H-pyrazol-4-yl)-4-{[4-methyl-3-oxo-2-(propan-2-yl)piperazin-1-yl]methyl}benzamide
(3S,4S)-4-methyl-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine-3,4-diol
2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-1,3-benzoxazole
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]pyridazine
4-(4-chlorophenyl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]butanamide
2-({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-[3-(dimethylamino)propyl]-N,2,5-trimethyl-1,3-thiazole-4-carboxamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
1-(2-methylpropyl)-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
8-[1-(4-chlorophenyl)cyclopropanecarbonyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}but-2-yn-1-one
4-propyl-1-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-5-one
{2-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-8-methylquinolin-3-yl}methanol
5-{imidazo[1,2-a]pyridine-3-carbonyl}-3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(2-hydroxyphenoxy)-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(quinoline-6-carbonyl)piperidine-3-carboxylate
(2S,4R)-4-(dimethylamino)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxylic acid
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(pyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-(3-methylbut-2-en-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
5-ethyl-N4-methyl-N4-[2-(morpholin-4-yl)propyl]pyrimidine-2,4-diamine
5-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(thiophen-2-yl)-1,2,4-oxadiazole
2-{6-[ethyl(methyl)amino]pyrimidin-4-yl}benzamide
1-(6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-yl)piperazine
N-cyclooctyl-2-{[2-(1H-indol-3-yl)ethyl]amino}acetamide
2-methyl-6-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-2,3-dihydropyridazin-3-one
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(pyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
methyl 1-[(3S,5S)-1-[(2-fluoro-4-methoxyphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[1-(2,7-dimethylquinoline-4-carbonyl)piperidin-4-yl]ethan-1-ol
(1R,9S)-5-amino-3-(4-fluoro-2-methylphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
N-[1-(2,5-difluorophenyl)cyclopropyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-({[(3R,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(2S)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
3-hydroxy-2-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]benzamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(3-methylphenoxy)piperidine
2-(azepan-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
N-cyclopentyl-N'-{2-[(4-methylpyridin-2-yl)amino]ethyl}butanediamide
6-(3-carbamoylpiperidin-1-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
N,2,6,8-tetramethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinoline-4-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-[3-(furan-2-yl)phenyl]urea
1-(cyclopropanesulfonyl)-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[(3S)-2-oxoazepan-3-yl]-1H-1,3-benzodiazole-7-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(4-methylphenyl)quinoline-4-carboxamide