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6-(2,5-dimethylfuran-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(4-fluoro-2-methylphenyl)-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
ethyl 1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(4aS,7aR)-1-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-methoxy-3-methylphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
(1S,5R)-3-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 3-[(3S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
N-[(2-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-2-(propan-2-yl)pyrimidine-5-carboxamide
1-ethyl-3-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-[2-(methylsulfanyl)phenyl]acetamide
3-(2,4-dimethoxybenzoyl)-1-[3-(methylsulfanyl)propyl]piperidine
N-methyl-6-oxo-N-[(4-phenoxyphenyl)methyl]-1,6-dihydropyrimidine-5-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)furan-2-carboxamide
2-methoxy-N,N-dimethyl-5-({[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzamide
N-cyclohexyl-N-[2-(dimethylamino)ethyl]-5-methyl-1,3-oxazole-4-carboxamide
1-(2-benzylmorpholin-4-yl)-3-(thiophen-2-yl)propan-1-one
methyl 2-({6-phenylimidazo[2,1-b][1,3]thiazol-3-yl}formamido)acetate
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
N-(oxan-4-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(pyridin-2-yl)ethyl]acetamide
(3R)-N-(3-butanamidophenyl)-3-hydroxypyrrolidine-1-carboxamide
6-[2-(3-methylphenyl)acetyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
6-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
dimethyl[2-(2-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenoxy)ethyl]amine
2-[1-(3-methylbutyl)-2,4-dioxo-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
2-[5-(azocan-1-ylmethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
6-methyl-2-({4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
N-cyclooctyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-ethyl-3-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]-N-phenylpropanamide
1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
3-fluoro-2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
(4aS,8aR)-6-{2-[benzyl(methyl)amino]acetyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
(7R,9aR)-7-methyl-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-ethyl-6-[4-(4-propylphenyl)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-indole-2-carboxamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
4-{4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
5-fluoro-2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-ethyl-N-methyl-3-({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}sulfamoyl)benzamide
4-(furan-2-carbonyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-benzyl-4-(3-hydroxypropyl)-1-(2-phenylphenyl)piperazin-2-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(hydroxymethyl)cyclopentyl]-3-{[(5-methylthiophen-2-yl)methyl]amino}benzamide
N-cyclopentyl-N-propyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrrole-2-carboxamide
N-[1-(6-methylpyridin-2-yl)propyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide