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[1-(5-{[1-(propan-2-yl)piperidin-4-yl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
8-[2-(morpholin-4-yl)pyridine-3-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1,3-dimethyl-5-(3,4,5-trimethoxyphenyl)-1H-1,2,4-triazole
2-ethoxy-5-{2-[3-(methoxymethyl)pyrrolidin-1-yl]pyrimidin-4-yl}benzoic acid
2-methoxy-N-[4-methyl-3-({[1-(pyrazin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]acetamide
2-(dimethylamino)-1-[4-(2-methoxyethyl)piperidin-1-yl]-2-(4-methylphenyl)ethan-1-one
1-(morpholin-4-yl)-3-[3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
4-{[1-(6-methylpyridin-3-yl)ethyl]amino}pyrimidine-5-carboxylic acid
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(piperidin-3-yl)benzamide
1-(2,5-di-tert-butylphenyl)-3-(2-oxopiperidin-3-yl)urea
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
3-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-5-(propan-2-yl)-1,2-oxazole
(3aS,6aR)-5-[(3,4-dimethylphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(4aS,7aR)-1-(3,5-difluoropyridine-2-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-methoxy-N,3-dimethylbenzamide
N-{2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
1-({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,4-diazepan-5-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
6-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(4aR,8aS)-1-(cyclohexylmethyl)-6-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-ethyl-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-methylpropan-1-one
2-methyl-N-(1-{1-[4-methyl-4-(methylsulfanyl)pentan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
methyl 4-(4-ethoxyphenyl)-1H-pyrrole-2-carboxylate
[(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
(1-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}ethyl)dimethylamine
4-({4-[4-methyl-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
5-[(4-benzylpiperidin-1-yl)methyl]-N-[1-(pyrimidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
(3R,4R)-4-ethyl-1-[2-(3-methylphenyl)benzoyl]piperidine-3,4-diol
1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperidine-4-carboxamide
6-(3-fluoro-4-methoxyphenyl)-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(2,4-difluorophenyl)-1-[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
(2R,3S,6R)-3-(4-methylphenyl)-5-[(2-propylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N,3,5-trimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-indole-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(3-methoxypropyl)amine
4-methyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-2-oxopentanamide
dimethyl(3-{2-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
5-ethyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1,3,4-oxadiazol-2-amine
3-[(2E)-2-methylpent-2-en-1-yl]-3,9-diazaspiro[5.5]undecane
3-(4H-1,2,4-triazol-4-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]benzamide
1-(3,5-dichloro-4-methylbenzoyl)-N,N-dimethylazepan-4-amine
1-methyl-4-phenyl-3-[1-(pyrimidine-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(3-chlorothiophene-2-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine