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(1R,5S,6S)-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carboxamide
1-(2,3-dimethoxyphenyl)-2-(4-methylbenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-phenyl-1H-pyrazole
9-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-{2-[3-(methanesulfonylmethyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
2-{2-oxo-8-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)-4-[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]pyrimidine
9-(2,6-dimethylpyridin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methylphenyl)-5-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
1-(4-methoxybenzoyl)-4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperazine
2-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-octahydropyrrolo[1,2-a]piperazine
methyl (2R,4S)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-4-hydroxypiperidine-2-carboxylate
4-{2-[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-amine
N-{2-methoxy-5-[(3E)-pent-3-enamido]phenyl}benzamide
methyl 4-({[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}carbamoyl)butanoate
2-[4-(2-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
methyl (2S,3S)-2-[(1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]phenyl}piperidin-4-yl)amino]-3-methylpentanoate
N-cyclopropyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-cyclopentyl-5-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(methylsulfanyl)-N-[2-(oxan-2-yl)ethyl]benzamide
methyl 5-(benzylamino)-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-(2-methylpropyl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)ethan-1-one
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-4-(pyrrolidin-1-yl)butan-1-one
N-[(2R,3R)-2-ethoxy-1'-[3-(1,2-oxazolidin-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-butyl-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carboxamide
3-(3,4-difluorophenyl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrazine
2-{2-[2-(4-chlorophenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-1-(piperazin-1-yl)ethan-1-one
2-(2-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
2-methoxy-1-(4-{4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
(2S,4R)-4-amino-1-[3-(1H-imidazol-2-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(2,3-difluorophenyl)methyl]acetamide
1-cyclopentyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
1-{2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]ethyl}imidazolidin-2-one
7-fluoro-3-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)-1,2-dihydroquinolin-2-one
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
8-(4-hydroxy-6-oxo-1-phenyl-1,6-dihydropyridazine-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-1,2,5-thiadiazole-3-carboxamide
1-(3-chlorophenyl)-4-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}piperazine
(3S,4S)-4-[4-(hydroxymethyl)piperidin-1-yl]-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-ol
2-[3-benzyl-1-(2-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-[(2R,3R)-1'-(2,3-dimethylbenzoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide