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1-(3-methoxyphenoxy)-3-({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)propan-2-ol
1-(2-methanesulfonylethyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
4-(quinolin-8-yl)phenol
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
1-(cyclopropylmethyl)-5-[2-(2,5-difluorophenyl)acetyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methoxy-6-[(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
N-cyclobutyl-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
(3S,5R)-N3-cyclopentyl-N5-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-(quinolin-2-ylmethyl)propanamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(3-methoxyphenyl)methyl]benzamide
1-(1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)pyrrolidin-2-one
4-{2-oxo-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethyl}-4-azatricyclo[4.3.1.13,8]undecan-5-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(2-ethylpyrimidin-4-yl)methyl]methylamine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-({[(3R,4R)-1-(2,6-dimethylpyridine-4-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-cyclobutyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(oxolane-3-carbonyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-(2-methoxyphenyl)-1H-pyrazole
methyl 7-oxo-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(4-phenylbenzoyl)-1-(1,3-thiazole-4-carbonyl)piperidine
N-benzyl-N-butyl-2-[1-cyclopropyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
2-({1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}oxy)pyrimidine
N-methyl-4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-2-amine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}benzonitrile
2-({[3-(2-methoxyphenoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
3-(3-methoxypropyl)-1-[(2-methylphenyl)methyl]piperidine-3-carboxylic acid
N-(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperidin-4-yl)acetamide
methyl 1-methoxy-2-oxo-8-(1-phenyl-1H-pyrazole-4-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(3-methyl-1,2-oxazol-5-yl)methyl](oxolan-2-ylmethyl)amine
3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4-(3-phenylpropyl)piperazin-2-one
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-{[5-(4-fluorophenyl)-4-[1-(pyridine-4-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
N-(2,4-dimethylphenyl)-3-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-oxopropanamide
1-phenyl-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazin-2-one
{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
N,N-diethyl-2-(4-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazine-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
4-[(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)methyl]morpholine
6-methoxy-3-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1-benzofuran-2-carboxamide
N,N-dimethyl-2-(pyridin-4-yl)-7-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N3-cyclooctyl-N5-(2-methoxyethyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-(hydroxymethyl)-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-6-methoxyquinolin-2-ol
5-methyl-6-(3-methylpiperidine-1-carbonyl)-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
3-(methylsulfanyl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]propanamide
(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
2-ethyl-9-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one