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7-[(4-fluorophenyl)methyl]-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
2-ethyl-9-(2-hydroxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-hydroxypropyl)-8-[(5-propylfuran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(6-chloro-2H-chromene-3-carbonyl)-3-(1H-imidazol-1-ylmethyl)piperidine
N-[2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
4-(methoxymethyl)-5-methyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1,2-oxazole-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1H-1,2,3-triazole-5-carboxamide
3-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,1-benzoxazole
2-(3-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-benzothiophene-5-carboxamide
N-({1-[(4-methanesulfonylphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-methylacetamide
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
(1r,4r)-4-{5-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}cyclohexan-1-ol
2-methoxy-N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-(cyclohexylmethyl)-N3-cyclopropyl-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)-1H-indole-7-carboxamide
2-benzoyl-6-methyl-5-[5-(1-methylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(carbamoylmethyl)-N-{[5-(4-fluorophenyl)furan-2-yl]methyl}piperidine-4-carboxamide
1-[(3-methylphenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
methyl 3-(oxolane-3-amido)-5-{[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-({2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-(4-ethyl-5-methylpyrimidin-2-yl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
(2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
N-[(4-fluoro-2-methoxyphenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
ethyl({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})(pyridin-4-ylmethyl)amine
3-(2,5-difluorobenzoyl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine
4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]thiomorpholine
9-(2,4-dimethylpyrimidine-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(4aR,7aS)-1-methyl-4-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3,4-dimethylphenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
(3R,4R)-1-[(2-hydroxynaphthalen-1-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-[(2R,3R,6R)-5-[4-(hydroxymethyl)benzoyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N3-cyclohexyl-N5-[1-(furan-2-yl)ethyl]-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-indole-6-carboxamide
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-amino-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-ethyl-1,3-thiazole-5-carboxamide
3-ethyl-8-[4-(1H-pyrazol-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N4-methyl-N4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-6-(pyrrolidin-1-yl)pyrimidine-2,4-diamine
5-(4-methyl-1,4-diazepan-1-yl)-2-(2-phenylethyl)-2,3-dihydropyridazin-3-one
(2S)-2-[(2-ethylpyrimidin-5-yl)formamido]-3-phenylpropanamide
3-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}imidazolidine-2,4-dione
6-{4-[3-(dimethylamino)-2,2-dimethylpropyl]piperazin-1-yl}pyridine-2-carbonitrile
1-(4-methoxybenzoyl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(thian-4-yl)piperazine
2-(1-{[4-(difluoromethoxy)phenyl]methyl}azetidin-3-yl)-1H-1,3-benzodiazole