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2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
2-({1-[(4-methylphenyl)amino]cyclopentyl}formamido)-N-(1,3-thiazol-2-yl)acetamide
5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-fluoro-2-methylphenyl)methyl]piperidine
4-[3-(azetidine-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
3-(1,3-thiazol-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(morpholin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[1-(pyrazin-2-yl)piperidin-4-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-benzyl-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}piperazin-1-yl)propanamide
(3aR,7aS)-2-(6-methoxypyrimidin-4-yl)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
[4-(3-phenylpropyl)-1-(pyrazin-2-yl)piperidin-4-yl]methanol
N,6-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
(2S)-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylamino)propanamide
N-(cyclopropylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(1,2,3-thiadiazol-5-yl)urea
N-{2-[1-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-[2-(dimethylamino)-4-{[2-methoxy-2-(thiophen-2-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-{5-[(3-methoxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-(1-{1-[(8-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
ethyl 1-ethyl-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazole
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(pyridin-3-yl)acetamide
5-acetyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]thiophene-3-carboxamide
(3E)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-phenylbut-3-enamide
N2,N2,6-trimethyl-N4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrimidine-2,4-diamine
2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(oxan-4-ylmethyl)acetamide
4-(1H-imidazol-2-yl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
N-methyl-4-(piperidin-1-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
1-ethyl-6-oxo-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(oxolan-3-ylmethyl)piperidine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(1,3-thiazol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[3-(methylsulfanyl)phenyl]ethan-1-one
2-(ethoxymethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
2-(dimethylamino)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-(3-methylphenyl)acetamide
2-{[(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-(2-methoxy-4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-(2-methoxyethyl)-N-methylacetamide
2-[3-(4-methyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
2-(1-methyl-1H-pyrazole-5-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-methoxy-6-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}phenol
3,5-dimethyl-2-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,4-dihydropyridin-4-one
{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
3-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]azetidin-3-yl}pyridine
[(2-ethylpyrimidin-5-yl)methyl](methyl){[1-(morpholin-4-yl)cyclohexyl]methyl}amine
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(4-methoxyphenyl)-2,2-dimethyl-N-(1,2-oxazol-3-ylmethyl)cyclopropane-1-carboxamide
4-[(4-fluorophenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1'-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol