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{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)[3-(1H-pyrazol-1-yl)propyl]amine
ethyl 4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
1-{[5-(1H-imidazol-2-yl)thiophen-2-yl]methyl}piperidine
4-(3-chloropyridin-2-yl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methylphenoxy)piperidine
(3S,4R)-1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-methylpiperidine-3,4-diol
1-{[5-(5-chloro-3-fluoropyridin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
5-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
N-cyclohexyl-N,5-dimethyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N,2,3,5-tetramethyl-N-[(3-methylpyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(pyrrolidin-1-ylmethyl)-1-(2,4,5-trimethylbenzoyl)piperidin-3-ol
1-[6-(3-methoxyphenyl)pyridine-3-carbonyl]-4-phenylazepane
5-(methoxymethyl)-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)furan-2-carboxamide
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
5-methyl-4-({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
(1R,5R)-6-(cyclopropylmethyl)-3-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-methyl-6-{3-[(methylsulfanyl)methyl]piperidin-1-yl}pyrimidin-2-amine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carboxamide
6-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine
N-[(3R,4S)-4-cyclopropyl-1-(3-methylbutanoyl)pyrrolidin-3-yl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
4-({[2-(azepan-1-yl)ethyl](propan-2-yl)amino}methyl)benzoic acid
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-methylimidazo[1,2-a]pyrimidine
5-{2-[(2-methylpiperidin-1-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-4-propylpyrimidine
1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
2-methyl-4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
N-(2-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoic acid
4-(4-propyl-1H-1,2,3-triazol-1-yl)-1-[4-(1H-pyrazol-5-yl)benzoyl]piperidine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(carbamoylmethyl)piperidin-4-yl]propanamide
1-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
2-({2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}sulfonyl)benzonitrile
1-(azocan-1-yl)-3-(2-methoxy-5-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
2-methyl-4-[4-(pyrrolidine-1-carbonyl)phenyl]-1H-imidazole
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-(3,4-dimethyl-1H-pyrazol-5-yl)propan-1-one
8-{3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-(2-methyl-1,3-thiazol-4-yl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)acetamide
7-hydroxy-6-methyl-4-[2-(propan-2-yl)pyrimidin-4-yl]-1,2,3,4-tetrahydroquinolin-2-one
6,8-dimethyl-3-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
8-(5-chloro-2-methylpyrimidine-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-({1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
1-(4-{[(2R,5S)-5-(1-benzofuran-5-ylmethyl)oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
4-hydroxy-2-phenyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
(3R,4R)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one