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(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2,1,3-benzoxadiazol-4-ylmethyl)({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
N-cyclohexyl-N-(pyridin-3-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-methyl-5-oxo-1-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,5-dihydro-1H-pyrazole-3-carboxamide
3-{2-[9-methoxy-7-oxo-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-3-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-methoxypropan-1-one
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-(1-ethyl-1H-pyrazol-4-yl)-6-methylquinoline
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(1-methoxybutan-2-yl)piperidine-4-carboxamide
1-(3-methylbutyl)-2-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
3-benzyl-1-methyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-chlorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
3-(2-{[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}ethyl)-1,3-oxazinan-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-(5-fluoro-2-methoxyphenyl)-2-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)acetic acid
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl][(1-phenyl-1H-pyrazol-4-yl)methyl]amine
N-{3-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
2-{3-oxo-3-[2-(pyridin-2-yl)piperidin-1-yl]propyl}-2,3-dihydro-1H-isoindol-1-one
8-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
4-(3-bromophenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(5-methylpyrazin-2-yl)methyl]-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
[(4-chloro-3-fluorophenyl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-phenylpyrimidine-5-carboxamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-2,5-dimethylfuran-3-carboxamide
3-[4-(3,4-dichlorobenzoyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
methyl 3-acetamido-1-(oxolan-2-ylmethyl)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-6-methyl-2-propylpyrimidine
methyl 2-{2-[2-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)acetamido]-1,3-thiazol-5-yl}acetate
1-[(4-methoxyphenyl)methyl]-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]pyridine-2-carbonitrile
(4aR,7aS)-1-ethyl-4-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
methyl 3-[2-(naphthalen-2-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-cyclobutyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methylpiperidin-3-amine
(3aS,6aS)-2-[(3-hydroxyphenyl)methyl]-5-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-methoxybenzoyl)-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
4-(2,6-dimethylpyrimidine-4-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)furan-2-carboxamide
2-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-{1-[1-(thiophen-2-yl)propyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
4,6-dimethyl-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide