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3-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
(3S,5S)-5-(morpholine-4-carbonyl)-1-(4-propylbenzoyl)piperidine-3-carboxylic acid
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-methylphenyl)propanamide
5-(2,6-difluorophenoxymethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
3-{5-[1-(1-benzylpyrrolidin-3-yl)-1H-1,2,3-triazol-4-yl]thiophen-3-yl}prop-2-yn-1-ol
(1S,5R)-N-[3-(methylsulfanyl)phenyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
[(3R,5R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
5-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylpyrimidin-4-amine
4-{2-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]quinolin-3-yl}butan-2-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-fluorophenyl)benzamide
1-(1-benzothiophene-2-carbonyl)-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
2-amino-N-[2-(2-chloro-6-methylphenoxy)ethyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
6-(cyclobutylamino)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-amino-6-(3-hydroxyphenyl)-4-(6-methoxy-2H-1,3-benzodioxol-5-yl)pyridine-3-carbonitrile
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-indole-6-carboxamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[(6-methylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(2S)-1-(5-phenyl-1,2-oxazole-4-carbonyl)pyrrolidine-2-carbonyl]morpholine
1-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)acetamide
1-[(2-fluorophenyl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-2-one
5-(3-chloro-4-methoxyphenyl)-2,3-dimethylpyrazine
3-(2-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
4-[(2-phenylpropyl)amino]-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
5-(3-phenylpiperazine-1-carbonyl)-2-(pyrrolidin-1-yl)pyrimidine
4-(2,4-dimethyl-3-oxopiperazine-1-carbonyl)benzene-1-sulfonamide
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-{[(2,3,4-trimethoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(1-ethyl-1H-indol-4-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
(3S,4R)-4-(4-fluorophenyl)-1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)pyrrolidine-3-carboxylic acid
3-(1-butyl-1H-pyrazol-5-yl)-1-[2-(4-sulfamoylphenyl)ethyl]urea
N-[4-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}methyl)phenyl]butanamide
4-(2-{1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethyl)-1,3-thiazol-2-amine
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-hydroxypropyl)acetamide
ethyl 5-(2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methyl-5-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
7-(oxan-4-yl)-2-(thiophen-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-fluorophenyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
2-(ethylamino)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
(9aR)-2-methyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1-methyl-1H-imidazol-2-yl)({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl})methanol
methyl 3-[(cyclohexylformamido)methyl]-5-(4-fluorobenzenesulfonamido)benzoate
3-(2,2-dimethyloxan-4-yl)-1-(4-ethoxy-2-fluorophenyl)-3-ethylurea
3-(5-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-(1-methyl-1H-imidazol-2-yl)-N-(2-phenylphenyl)piperidine-1-carboxamide
1-(2-{[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)imidazolidin-2-one