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4-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3-ethylpiperazin-2-one
2-methyl-N-{[3-methyl-7-(5-phenoxyfuran-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-4-carboxamide
(4aS,7aR)-1-[(2-fluorophenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-4-methylbenzene-1-sulfonamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
1-(pyridin-4-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4-diazepane
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-hydroxypiperidin-1-yl)acetamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
4-[(2-methylphenyl)methyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
2-(3-fluorophenoxymethyl)-N-(3-hydroxy-3-methylbutyl)-N-methyl-1,3-oxazole-4-carboxamide
(2S)-2-{3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanamido}-3-phenylpropanoic acid
2-{9-[(5-fluoro-2-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
2-cyclopentyl-1-[4-(2-methoxy-5-{[methyl(propan-2-yl)amino]methyl}phenoxy)piperidin-1-yl]-2-phenylethan-1-one
1-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidin-3-ol
N-(2-hydroxyethyl)-3-{5-[(trimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
ethyl (4aR,6R,8aS)-2-(furan-2-ylmethyl)-6-(morpholin-4-yl)-decahydroisoquinoline-8a-carboxylate
2-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(1H-pyrrol-1-yl)propanamide
4-[2-chloro-4-(cyclopentylcarbamoyl)phenoxy]-N,N-dimethylpiperidine-1-carboxamide
2-{4-[(2,5-dimethylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-(cyclopropylmethyl)-9-[2-(4-fluoro-3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,4-dioxan-2-ylmethyl)-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
N-cyclopentyl-2,3-dimethoxy-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
2,5-dimethyl-3-[3-(pyridin-4-yl)azetidin-1-yl]pyrazine
3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-(2-methyl-1H-1,3-benzodiazol-6-yl)urea
(1R,5S,6S)-6-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
(2S,4R)-4-amino-N,N-diethyl-1-(1-ethyl-1H-pyrazole-3-carbonyl)pyrrolidine-2-carboxamide
(3S,4R)-1-[3-(dimethylamino)propanoyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[3-(2-fluorophenyl)benzoyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
(3R,9aR)-3-(2-methylpropyl)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
6-fluoro-4-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinolin-2-one
1-(2,5-difluorobenzoyl)-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
5-(methoxymethyl)-N-[4-(5-methyl-4-{[2-(pyridin-3-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]thiophene-2-carboxamide
N4-(1-phenylcyclopropyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
[(3R,4R)-1-(5-methoxyfuran-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-cyclopropyl-1-(5-phenoxyfuran-2-carbonyl)piperazine-2-carboxamide
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-2-[4-(prop-2-en-1-yl)piperazin-1-yl]pyrimidine
N4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N2,N2,N4-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(1R,2S)-N1-tert-butyl-N2-(2-methanesulfonylethyl)cyclohexane-1,2-dicarboxamide
ethyl 3-benzyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
(1R,3S)-7-(3-chloropyridin-2-yl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
4-[2-(5-methylfuran-2-yl)phenyl]-4H-1,2,4-triazole
4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(propan-2-yloxy)ethyl]benzamide
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
5-(5-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
3-tert-butyl-1-[1-(pyridine-3-sulfonyl)azepan-3-yl]urea
methyl N-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}carbamate
2-(1H-1,2,3-benzotriazole-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one