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methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{1-[2-(2,3-difluorophenyl)acetyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
(2S,4R)-N-[3-(2-ethylphenoxy)propyl]-4-hydroxy-N-methylpyrrolidine-2-carboxamide
5-({1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl}methyl)-1,2-dihydropyridin-2-one
1-(methoxymethyl)-N-[(4-methoxynaphthalen-1-yl)methyl]-N-methylcyclobutane-1-carboxamide
N-[2-(ethylsulfanyl)phenyl]-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
2-cyclopropyl-N,N-dimethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
3,4,4-trimethyl-1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-3-ol
[5-({cyclohexyl[2-(ethylsulfanyl)ethyl]amino}methyl)furan-2-yl]methanol
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
3-{4-[3-(pyridin-2-yl)azetidine-1-carbonyl]piperidin-1-yl}-1λ6-thiolane-1,1-dione
4-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-ethyl-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
methyl N-{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoethyl}carbamate
N-(furan-2-ylmethyl)-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)pyridine-3-carboxamide
2-[(1S,5R)-3-(3,5-dimethoxybenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[3-(4-fluorophenyl)propyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-ethyl-N,4-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazole-5-carboxamide
3-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
{[2-(4-ethylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}(1-methoxypropan-2-yl)amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
[1-(3-methylpyridin-2-yl)propan-2-yl]({1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
methyl 3-acetamido-5-{[1-(2-fluorophenyl)propan-2-yl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-dihydroquinolin-2-one
1-cyclopentyl-3-{2-[4-(2,5-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)pyrrolidine-2,5-dione
8-(2,5-dichlorobenzenesulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-{[(5-fluoro-2-hydroxyphenyl)methyl](methyl)amino}-N,2-dimethylpropanamide
5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazole
2-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepan-5-one
4-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-[(3,5-difluorophenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-methyl-4-{[propyl(pyridin-3-ylmethyl)amino]methyl}benzene-1-sulfonamide
(1R,6S)-N-cyclopentyl-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-fluoro-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}benzamide
N-[(2R,3R)-1'-(2H-1,3-benzodioxol-5-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
N-[3-(dimethylamino)propyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-methyl-1-(2-methylpropyl)-4-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-[2-(1H-imidazol-2-yl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
ethyl 2-[4-(4-amino-5-cyanopyrimidin-2-yl)piperazin-1-yl]acetate
N-[2-(furan-2-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
2-methoxy-3-(4-methylpyridin-3-yl)quinoline
1-cyclopentyl-3-(2-fluorophenyl)-3-{2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
4-[2-(4-{2-[4-(methylsulfanyl)phenyl]acetyl}morpholin-3-yl)acetyl]piperazin-2-one
2-{2-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
2-(2-{[cycloheptyl(ethyl)amino]methyl}phenyl)-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
methyl (2S,4S)-1-(1-benzylpiperidin-4-yl)-4-(2-methylquinoline-4-amido)pyrrolidine-2-carboxylate
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}piperidin-4-amine