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(4aS,7aR)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-1-(3,5-dimethylphenyl)piperazin-2-one
(1S,5R)-3-(pyridine-2-carbonyl)-6-(2,2,3,3-tetramethylcyclopropanecarbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-fluoro-2-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-methylquinoline
N-[(4-methoxyphenyl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-methyl-3-phenylpiperidine
(4aS,8aR)-1-(carboxymethyl)-6-[(2,3-difluorophenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
6-oxo-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
6-methyl-N4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
N-[2-(1-{2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetyl}piperidin-4-yl)ethyl]acetamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)piperidin-2-one
4-[2-(2-fluorophenyl)ethyl]-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
7-methyl-2-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2,3-dihydro-1H-inden-2-yl)-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazole
3-(2-methoxyethyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidine-3-carboxylic acid
N-(2-methoxyethyl)-3-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}propanamide
1-cycloheptyl-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
N-cyclopentyl-N-[(2,4-dimethoxyphenyl)methyl]-1,5-dimethyl-1H-pyrazole-4-carboxamide
2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-6-(2-methoxyphenyl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyridine-3-carboxamide
2-cyclopropyl-1-{6-methyl-5-[5-(pyridazin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
N-{[1-(2-acetylbenzoyl)piperidin-3-yl]methyl}-4-phenylbenzamide
1-[(3,5-dichloropyridin-4-yl)methyl]-4-(2-phenoxyethyl)piperazine
3-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}pyridine
3-benzyl-4-[4-(1H-pyrrol-1-yl)benzoyl]piperazin-2-one
1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-4-phenylpiperidine-4-carbonitrile
6-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(3-methylpyridin-4-yl)piperazine
3,5-dimethyl-4-{2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propyl}-1H-pyrazole
1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(furan-3-yl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-3-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)quinolin-8-amine
2-[(3,4-difluorophenyl)methyl]-8-(3-hydroxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(2-chlorophenyl)-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
11-{[(2,5-difluorophenyl)methyl]amino}-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-9-[4-(propan-2-yl)benzenesulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
8-cyclohexyl-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl (2S)-1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
11-{[(4-fluorophenyl)methyl]amino}-4-[2-(2-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl (2R,4S)-4-hydroxy-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidine-2-carboxylate
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-methyl-1-[(5-methylfuran-2-yl)methyl]urea
methyl 9-[(4-fluorophenyl)methoxy]-3-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
3-[4-(2-fluoro-3-methylphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
2-{[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one