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2-({[(2,4-dimethoxyphenyl)methyl]amino}methyl)-6-fluoroquinolin-4-ol
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(pyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-chloro-N-[2-(2,5-dimethylphenoxy)ethyl]-N-methylpyridine-4-carboxamide
1-(3-{[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-2,4,6-trimethylphenyl)ethan-1-one
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
1-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine
6-(3-chlorophenyl)-N-(2,3-dihydroxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[4-(methylsulfanyl)phenyl]ethan-1-one
ethyl 1-(3-methylfuran-2-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5,6-dimethylpyrimidin-4-amine
4-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1-methylpiperazin-2-one
3-fluoro-5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]benzonitrile
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(3-methoxyphenyl)propanoyl]piperidine-3-carboxylate
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
(3S,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4-phenyl-1,2,3-thiadiazol-5-yl)pyrrolidine-1-carboxamide
N-{4-chloro-3-[({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}carbamoyl)amino]phenyl}-2-methoxyacetamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
9-hydroxy-2-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
5-ethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-4H-chromen-4-one
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(2,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-3-yl)prop-2-enamide
6-[4-(2-fluorophenyl)benzoyl]-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
[(5-{1-[(2,3-difluoro-4-methylphenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
methyl 2-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}amino)acetate
3,4-difluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
1-ethyl-3-(morpholine-4-carbonyl)-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
6-({[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}methyl)-1,4-oxazepan-6-ol
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-(2-fluorobenzoyl)pyrrolidine-2-carboxamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
8-pentanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazine
3-[(pyridin-2-ylmethyl)sulfamoyl]-5-(pyridin-4-yl)benzoic acid
[5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-2-(propan-2-yloxy)phenyl]methanol
3-[(furan-2-ylformamido)methyl]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
N-cyclohexyl-1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-(3,5-dimethylphenyl)-N'-methyl-N'-[1-(pyridin-4-yl)ethyl]propanediamide
5-cyclopropyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-1,3,4-oxadiazol-2-amine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]quinoxaline-5-carboxamide
N-(3-hydroxypropyl)-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-(2-ethylbutanoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[1'-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one