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2-[4-(piperidine-1-carbonyl)phenyl]pyrazine
(2S)-3-methyl-2-(3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)butanamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-indole
(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
(2S,4R)-4-amino-1-(4-chloro-2-methylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(2,3-difluorophenyl)methyl]-4-[1-(3-methylfuran-2-carbonyl)pyrrolidin-3-yl]piperidine
7-(5-chloro-2-ethoxyphenyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
1-[(4-fluorophenyl)methyl]-4-{[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]amino}pyrrolidin-2-one
1-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)-2-methylpiperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylfuran-3-carboxamide
5-ethyl-4-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-oxazole
methyl 1-[(3R,5S)-1-[(3-fluorophenyl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
9-(4-amino-3-hydroxybutanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(4-hydroxyphenyl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
(2S,4S)-4-amino-N-methyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
methyl 7-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-methyl-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-2-amine
5-cyclobutanecarbonyl-1'-(1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(4aR,7aS)-4-(3-methoxypropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(3R,4S)-1-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
N5-benzyl-N6-(propan-2-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-methoxypyrazine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-{2-[4-(3-cyclopentylpropanoyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-amine
N,N-dimethyl-2-phenyl-2-[(3-propyl-1H-pyrazol-5-yl)formamido]acetamide
N-(1-methoxypropan-2-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
{2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}urea
2-{1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-imidazole-4-carboxamide
5,7-dimethyl-3-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyrazolo[1,5-a]pyrimidine
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[1-(6-methylpyridin-2-yl)propyl]acetamide
(3R,9aR)-8-(2-methoxybenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[2-(2,6-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]benzamide
(1R,2R,6S,7S)-4-(2-methoxypyridine-3-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-[(4-hydroxy-3,5-dimethylphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1,2-oxazol-5-ylmethyl)acetamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
[(3R,4R)-1-(2-methylpyrimidine-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[(3S,4S)-3-hydroxy-4-(thiomorpholin-4-yl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-(piperidin-1-ylmethyl)benzamide
5-methyl-2-phenyl-N-[1-(thiophen-2-yl)ethyl]-1H-imidazole-4-carboxamide
3-(2-methoxyethyl)-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-{[(2R,3R)-3-[ethyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}pyridin-1-ium-1-olate
4-(1,3-benzothiazol-2-ylmethyl)-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine