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8-(1-benzofuran-2-ylmethyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
4-(1-{1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}ethyl)morpholine
4-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-(pyridin-2-yl)acetamide
1-(2-ethylpyrimidine-5-carbonyl)-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
(3R,4R)-1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-(3-{4-[5-(oxan-2-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}propyl)pyrrolidin-2-one
1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
[(3,5-dimethyl-1H-indol-2-yl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-(2H-1,3-benzodioxol-5-yl)-1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propan-1-one
1-(2-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
2,3-dimethoxy-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-3-carboxamide
1-[benzyl(methyl)amino]-3-(5-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]methyl}-N-[(5-methylfuran-2-yl)methyl]quinazolin-4-amine
2-amino-7-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4-benzyl-1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)methanol
N-(cyclopropylmethyl)-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
N-[1-(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
3-(2-ethylbutanamido)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methylbenzamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-(butan-2-ylsulfanyl)-5-(4-phenyl-1H-imidazol-5-yl)pyrimidine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-5-carboxamide
(4aS,7aR)-1-(pyridin-2-ylmethyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}benzamide
2-chloro-4-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}phenol
(1S,5R)-3-[6-(propan-2-yl)pyrimidin-4-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(dimethyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-{[7-(2-chloro-6-fluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
1-[3-(2-methoxyethoxy)phenyl]-3-(1-phenylcyclopropyl)urea
N-[4-({[(3S)-2-oxoazepan-3-yl]carbamoyl}methyl)phenyl]butanamide
5-(2-chloro-4-methoxyphenoxymethyl)-3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-pyrazole
1-{1-[1-(3-chloro-4-methoxybenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
methyl 4-[(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}quinazolin-4-yl)amino]butanoate
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(2-methylpropyl)-1,4-diazepan-1-yl]ethan-1-one
N-(4-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}phenyl)acetamide
(2H-1,3-benzodioxol-5-ylmethyl)({[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl})methylamine
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-3-yl)piperidin-4-ol
1-ethyl-3-methyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{4-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]piperidin-1-yl}-2-(propan-2-yl)pyrimidin-4-ol
2-{2-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
N-(1-benzylpyrrolidin-3-yl)-5-phenyl-1,2,4-triazin-3-amine
1-({4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
2-({[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(benzyl)amino)ethan-1-ol
N-methyl-N-[(4-phenoxyphenyl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide