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1-[1-(cyclopropylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-(3,4-difluorophenyl)-3-(2-methylpropyl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-(propan-2-yl)pyridazin-3-amine
methyl 5-[(2,2-dimethylpropyl)amino]-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
7-(1-benzothiophen-3-yl)-9-ethoxy-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[2-(1-methyl-1H-pyrazol-5-yl)ethyl]sulfamoyl}-N-(2-methylpropyl)benzamide
2-{3-[2-(methylsulfanyl)ethyl]-5-(4-oxo-1,4-dihydroquinolin-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
2-(2-butylpyrimidin-5-yl)-6-chloro-N,N-dimethylquinoline-4-carboxamide
N-(furan-2-ylmethyl)-3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-1-carboxamide
1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(propan-2-yloxy)ethan-1-one
[(1S,3S,3aS,6aR)-5-ethyl-3-[5-(hydroxymethyl)furan-2-yl]-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N4-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N4-methyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
6-(2-hydroxyethyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
3-({4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridin-2-amine
(4aS,7aR)-1-[2-(furan-2-yl)-2-oxoacetyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 3-(4-methoxybenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-ethyl-4-[2-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)ethyl]piperazine
2,5-dimethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-methoxyethyl)-4-methyl-3-({methyl[(methylcarbamoyl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
4,4-difluoro-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine
propan-2-yl N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]carbamate
N-[(3R,5S)-1-cyclopentanecarbonyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[4-(1H-pyrazol-4-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
methyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
4-(4-chloro-2-fluorophenyl)-5-[3-(methylsulfanyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine
4-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-2-methoxyphenol
4-[4-(piperazine-1-carbonyl)benzenesulfonyl]-1,4-oxazepane
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-[ethyl(methyl)amino]ethan-1-one
N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(pyridin-3-ylmethyl)acetamide
4-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]-N,N-dimethylbutanamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
5-(5-methylfuran-2-yl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1,2,4-triazin-3-amine
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[4-(propan-2-yloxy)benzoyl]pyrrolidin-3-yl]methanol
5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-(4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
1,3-dimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-(benzyloxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
5-(cyclopentylamino)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-ethyl-N-[2-(2-methylpropanesulfonyl)ethyl]pyrimidin-2-amine
N-(6-ethylpyridin-2-yl)-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{[4-(propan-2-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane