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ethyl 2-({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)amino)acetate
5-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
1-(cyclohex-3-en-1-ylmethyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
5-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
5-(3-fluorophenoxymethyl)-N-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
3-(oxolan-3-yl)-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazole
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
1-(3-{3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}propyl)piperidine
N-[(2-methoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[({1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-3-yl}oxy)methyl]pyridine
2-(dimethyl-1,3-thiazol-5-yl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-[1-(1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)ethyl]morpholine
3-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[4-(trifluoromethyl)phenyl]urea
N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
(3S,4S)-N-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-4-(dimethylamino)-3-hydroxypiperidine-1-carboxamide
1-({3-[(3-chlorophenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}methyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
3-[3-(2-hydroxyphenyl)propanamido]-4-(2-methylpiperidin-1-yl)benzamide
2-benzyl-N-ethyl-1-methyl-N-(oxolan-2-ylmethyl)-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
2-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}pyrazine
1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
4-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
N-benzyl-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
N-[1-({[2-methoxy-2-(thiophen-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
N3,N3-diethyl-1-(2-methoxyethyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-butyl-4-(1H-imidazol-4-ylmethyl)-1-(2-methoxyphenyl)piperazin-2-one
N-[2-(3-methoxyphenyl)-1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazin-2-one
4-[(2-ethylpyrimidin-4-yl)methyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane
2-[4-methyl-6-({1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}amino)pyrimidin-2-yl]phenol
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N4-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-6-methylpyrimidine-2,4-diamine
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
4-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-2-methylbutan-2-ol
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-propylacetamide
N4-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
4-(3-chloro-4-hydroxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-3-ethyl-5-methyl-1,2-oxazole
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
4-[2-amino-3-cyano-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]benzoic acid
N-[(2R,3R)-1'-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
2-[4-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)morpholin-3-yl]acetic acid
3-(4-benzyl-1H-pyrazol-5-yl)-1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
N-benzyl-5-(2-methoxyacetamido)-N,1-dimethyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
6,7-dimethoxy-4-(piperidin-1-yl)-2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}quinazoline
2-{1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1-oxobutan-2-yl}-2,3-dihydro-1H-isoindol-1-one
2-methyl-5-(propan-2-yl)-N-[2-(pyridin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-cyclohexyl-5-(2-fluoro-6-methoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole