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{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(ethyl)(2-methoxyethyl)amine
9-[(2-chloro-5-fluorophenyl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(2-hydroxyphenyl)propanamide
2-{1-cyclopentyl-4-[(8-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
7-[(5-methoxy-1H-indazol-3-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
5-benzamido-1-cyclopentyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
(2S)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(methylamino)hexan-1-one
1-{3-[2-(3-hydroxyphenyl)pyridin-4-yl]pyrrolidin-1-yl}-3-(pyridin-3-yl)propan-1-one
3-{2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]phenyl}pyrrolidine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
3-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-N-propyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethylpiperidin-4-amine
N-[3-(4-{[(2S)-2-acetamido-4-(methylsulfanyl)butanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]benzamide
2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(2-hydroxyethyl)acetamide
1-[2-(1H-imidazol-1-yl)acetyl]-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
(1S,5R)-3-[2-(ethylamino)pyrimidine-5-carbonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]piperazine-2-carboxylic acid
2-(5-ethyl-1-benzofuran-3-yl)-1-(6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
N-{2-[3-(1,2-oxazolidin-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
4-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
7-(3-chlorophenyl)-4-(9H-purin-6-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-methyl-N4-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrimidine-2,4-diamine
(4aS,8aS)-N-cyclohexyl-4a-hydroxy-7-(pyrazin-2-yl)-decahydro-2,7-naphthyridine-2-carboxamide
(furan-3-ylmethyl)(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amine
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)quinoxaline-5-carboxamide
4-[(4aS,7aR)-4-(3-methylbut-2-en-1-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
N-[4-({7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenyl]acetamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-(piperidin-1-ylmethyl)piperidin-2-one
N-(cyclohex-1-en-1-ylmethyl)-3-[(oxolan-3-yl)sulfamoyl]benzamide
5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1-cycloheptylpiperidin-2-one
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(1-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-1-oxobutan-2-yl)-2,3-dihydro-1H-isoindol-1-one
1-(4-chlorophenyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclopropane-1-carboxamide
3-{1-[2-(3-hydroxypiperidin-1-yl)acetyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
2-(3-methyl-1H-pyrazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2,3-dihydro-1H-inden-1-one
1-(carbamoylmethyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)piperidine
3-{5-[1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-2-yl]thiophen-3-yl}prop-2-yn-1-ol
5-tert-butyl-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-1,3,4-oxadiazol-2-amine
2-(2,4-dichlorophenoxy)-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-(furan-2-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one