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5-methyl-1-(2-methylphenyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
2-{4-[6-amino-5-cyano-4-(3-hydroxyphenyl)pyridin-2-yl]phenoxy}acetic acid
5-{[4-(5-ethylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{4-[(2,5-dimethoxyphenyl)methyl]piperazine-1-carbonyl}-1-methylazepane
N-[(2S)-1-cyclohexyl-3-hydroxypropan-2-yl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
methyl 3-{[3-(3-chlorobenzoyl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
5-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydropyridin-2-one
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-[3-(trifluoromethyl)phenyl]ethan-1-ol
{[4-(4-ethyl-3,3-dimethylpiperazine-1-carbonyl)-1,3-thiazol-2-yl]methyl}dimethylamine
1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-({[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)-6-methyl-3,4-dihydropyrimidin-4-one
3-[2-(3-fluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
1-[(4-ethylphenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylpiperidine-1-sulfonamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
(3S,4R)-1-cyclopentyl-4-phenylpyrrolidine-3-carboxylic acid
2-(2-hydroxyethyl)-8-(4-methoxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-6-(2,6-dimethylpyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-[1-(3-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
N-cyclohexyl-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(prop-2-yn-1-yl)propanamide
N-[2-(2-fluorophenyl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(3S,9aR)-3-(2-methylpropyl)-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
3-[1-(cyclopropylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
1-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-[(2,6-difluorophenyl)methyl]-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
(3S,4R)-4-(4-fluorophenyl)-1-[2-(1H-indol-3-yl)acetyl]pyrrolidine-3-carboxylic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-hydroxy-N-(1,2,3-thiadiazol-5-yl)-4-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1-[4-(4-ethylpiperazin-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
ethyl 4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-(1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
(3aS,6aS)-2-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-5,6-dimethylpyrimidine
6-ethyl-1,5-dimethyl-3-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydropyridin-2-one
4-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
3-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(3S)-N,N-dimethyl-1-(quinoxaline-5-carbonyl)azepan-3-amine
N-benzyl-3-(1-methylpiperidin-4-yl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
5-{1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}-N-cyclobutylthiophene-2-carboxamide
N-[2-(1-methylpiperidin-3-yl)ethyl]naphthalene-1-carboxamide
5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-[1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazol-4-yl)-N-methylformamido]-N,2-dimethylpropanamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-(2-methylbutyl)piperidine-4-carboxylate
1-[2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-2-methyl-1,4-dihydroquinolin-4-one
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(5-{1-[2-(2-hydroxyethoxy)ethyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol