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1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-methylphenoxy)piperidine
9-[(3S)-3-hydroxy-3-phenylpropyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-4-yl}-1-methyl-1H-1,3-benzodiazole
9-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1,4,9-triazaspiro[5.5]undecan-5-one
5-(cyclohex-3-en-1-yl)-1-ethyl-1H,4H-pyrazolo[3,4-d]imidazole
3-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-{1-oxaspiro[4.4]nonan-3-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-(2-oxoazepan-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-4-amine
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
N-ethyl-2-(4-hydroxyphenyl)benzamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
4-({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)-1-(3-phenylpropyl)pyrrolidin-2-one
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
2-{2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S)-1-[9-methoxy-3-(3-methylbenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
2-methyl-8-[3-(5-methylfuran-2-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(2E)-hex-2-en-1-yl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
3-pentanamido-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
N-{4-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethoxy]phenyl}propanamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]thiophene-2-carboxamide
1-(3-chlorophenyl)-5-methyl-3-(oxolan-3-yl)-1H-1,2,4-triazole
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[1-(3-methylpyridin-2-yl)propan-2-yl]amine
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
(1S,6R)-9-[1-(benzenesulfonyl)cyclopropanecarbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,1-benzoxazole-3-carboxamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(2-methoxyphenyl)propan-1-one
5,5-dimethyl-3-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidine-2,4-dione
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl})[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
6-cyclopentyl-N,1-dimethyl-N-[3-(pyrrolidin-1-yl)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-fluorophenyl)ethan-1-one
(3R,5S)-N3-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
2-methoxy-N-[2-(1,2,3-thiadiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
1-{4-[(1-hydroxypropan-2-yl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(4-{[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
(3aR,6aS)-5-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
N-[(2-methoxyphenyl)methyl]-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetamide
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
1-[(5-chlorothiophen-2-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[(E)-2-phenylethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(2S,4R)-N-methyl-4-{[(3-methylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
7-[(4-fluorophenyl)methyl]-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(6-chloropyridin-3-yl)methyl]-N,1,6-trimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide