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4-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]-1-(3,5-dimethylphenyl)piperazin-2-one
5-phenoxy-N-[2-(1H-pyrazol-4-yl)ethyl]furan-2-carboxamide
2-[4-(3-cyclohexyl-1H-pyrazol-4-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(3-methylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(pyridin-2-yl)propanoyl]pyrrolidine-2-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridine-4-carbonyl)piperidin-3-ol
5-(3-ethoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-(2-methoxyethyl)-2,6-dimethyl-N-(oxolan-2-ylmethyl)quinoline-3-carboxamide
1-cyclohexanecarbonyl-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
N-[(4-ethylphenyl)methyl]-4-hydroxy-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
8-methoxy-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(4-chlorophenyl)-3-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
2-chloro-6-methoxy-4-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
(4aR,7aS)-1-methyl-4-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2,3-dihydro-1H-inden-2-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-amine
1-(2-methanesulfonylethyl)-4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazine
1-methyl-5-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-benzotriazole
2-oxo-1-phenyl-N-[(1-phenylcyclopentyl)methyl]pyrrolidine-3-carboxamide
2-(dimethylamino)-1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]ethan-1-one
N-[(2R,3R)-1'-(2,3-dimethoxybenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-[(2-methoxyethyl)(methyl)amino]-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
8-(ethanesulfonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,7S)-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
8-(1-ethyl-1H-pyrazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylfuran-3-carboxamide
{5-[1-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]furan-2-yl}methanol
N,N-dimethyl-3-[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})sulfamoyl]benzamide
1-{2-[3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydroquinazolin-2-one
1-{4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}ethan-1-one
1-{[3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
(3S,4R)-1-[3-(methylsulfanyl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-amino-4-cyclopropyl-6-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridine-3-carbonitrile
3-{1-oxa-7-azaspiro[3.5]nonane-7-sulfonyl}-N-(oxolan-3-yl)benzamide
N-methyl-2-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-oxaspiro[4.5]decane-4-carboxamide
5-acetyl-N-[(2-methoxyphenyl)methyl]-6-methyl-2-oxo-N-propyl-1,2-dihydropyridine-3-carboxamide
3-{[(1-ethyl-3-methylpiperidin-3-yl)formamido]methyl}benzoic acid
2-(4-methoxy-3-methylphenyl)-5-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-3-(3-fluorophenyl)benzamide
2-(1,3-dimethyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-methyl-3-propyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide