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(1R,5R)-6-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[4-methyl-5-({1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)-4H-1,2,4-triazol-3-yl]methanol
1-ethyl-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]sulfonyl}piperazine
2-{5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}-1H-1,3-benzodiazole-6-carboxylic acid
3-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-yl)-1,3-oxazolidin-2-one
5-(3-phenylpropyl)-5-(piperidin-4-yl)-3-[2-(1H-pyrazol-1-yl)ethyl]imidazolidine-2,4-dione
(2E)-N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(pyridin-4-yl)prop-2-enamide
7-methyl-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-indole
4-{[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]amino}pyrimidine-5-carboxylic acid
(3R,4R)-1-(1-benzoylpiperidin-4-yl)-4-cyclobutyl-3-methylpiperidin-4-ol
3-methyl-1-(3-methylbutyl)-4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S)-1-benzyl-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidine
2-{3-[1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1H-pyrrole-3-carbonyl)piperidine
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
3-[(4-methoxypiperidin-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
methyl (2R,4S)-4-hydroxy-1-[4-methyl-3-(3-methylbutanamido)benzoyl]piperidine-2-carboxylate
3-[N-methyl-1-(3,5,7-trimethyl-1H-indol-2-yl)formamido]-3-phenylpropanoic acid
(3aR,6aS)-2-ethyl-1-oxo-5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
6-[4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-9H-purine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(4-methylphenoxy)acetamide
N-benzyl-2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-6-methylpyridine-3-carboxylic acid
2-[3-(2-ethoxypyridin-3-yl)-4-methoxyphenyl]ethan-1-amine
(1R,9S)-5-amino-3-(3-ethenylphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
4-[(dimethylamino)methyl]-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]azepan-4-ol
3-(6,7-dimethoxy-4-methylquinolin-2-yl)propanamide
2-(cyclopropylmethyl)-9-(2-methoxy-6-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohexylmethyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(1-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-(2-methoxyphenoxy)-2-methylpropan-1-one
1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
4-{1-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-4-phenyl-1H-imidazol-5-yl}-2-methoxyphenol
5-methyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-indole-2-carboxamide
8-[2-(dimethylamino)benzoyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(8-{[4-(diethylamino)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
9-methoxy-3-(3-methylbut-2-en-1-yl)-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidine
2-(2-fluorophenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-3-amine
1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(2-methylphenoxy)piperidine-4-carboxylic acid
N-{1-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxybenzamide
2-(4-phenyloxan-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-cyclopropyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzoxazole-6-carboxamide
6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
2-[1-methyl-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-yl]ethan-1-ol
5-cyclohexaneamido-N-[(3-fluoro-4-methylphenyl)methyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide