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2-benzyl-1-methyl-5-propanamido-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N,N-dimethyl-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)azepan-4-amine
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(pyridin-2-yl)piperidin-4-ol
N-[2-(2-fluorophenoxy)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-methyl-2,3,4,9-tetrahydro-1H-carbazole
2-(2-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-1H-1,3-benzodiazole
4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}piperidine-4-carboxylic acid
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2,2-dimethylpropyl 2,7-diazaspiro[4.5]decane-2-carboxylate
N-[4-(methylsulfanyl)phenyl]-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}acetamide
2-(3-fluorophenyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,3-benzoxazole-5-carboxamide
7-(3-chlorophenyl)-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[1'-(3-methoxypyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[3-(3-chlorophenyl)phenyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-4-carboxamide
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2-fluoro-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-5-sulfamoylbenzamide
(3aR,6aR)-2-benzyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-ethyl-5-{[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-(1-ethyl-3-methylpiperidine-3-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
[2-(furan-2-yl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(4aR,7aS)-1-(2-methoxyethyl)-4-[(3-methylquinoxalin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[(3R,4R)-1-[1-(4-fluorophenyl)piperidin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-4-(thiophen-2-yl)butan-1-one
(3R,5S)-N3-cycloheptyl-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
3-(propan-2-yl)-1-{[1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]methyl}urea
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(pyrazin-2-yl)propan-1-one
4-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}benzoic acid
N-cyclopropyl-2-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyridine-4-carboxamide
8-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
N-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
N-[1-(1H-indol-2-yl)ethyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
N-methyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,3-thiazol-2-amine
4-[(dimethylsulfamoyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-[5-(2H-1,3-benzodioxol-5-yl)-3-(2-ethoxyethyl)-1H-1,2,4-triazol-1-yl]-6-methylpyridine
3-{[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]sulfamoyl}-N-cyclopentylbenzamide
N-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
3-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
N-cyclopropyl-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-[2-(2-fluorophenyl)ethyl]-1-methylpiperidine
1-(cyclopropylmethyl)-5-(ethanesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(1H-imidazol-1-yl)ethyl]-3-(4-methylphenyl)-3-phenylpropanamide
N-{2-[5-(2-methoxypyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methylbenzamide
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyrrolidine-1-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2,6-dimethoxypyridine-3-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine