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1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine
4-[2-(3,4-dimethylphenoxy)ethyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-amine
N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(1S,4S)-2-(3-chlorophenyl)-5-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-(quinolin-8-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1,3-benzothiazole-6-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(2,6-difluoro-3-methylphenyl)methyl]amino}piperidin-1-yl)benzamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-cyclopentyl-N5-(2,3-dihydro-1H-inden-2-yl)-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(oxolan-2-ylmethyl)-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N,N-diethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
N-{1-[2-(aminomethyl)morpholine-4-carbonyl]cyclopentyl}-4-methoxyaniline
N-(3-hydroxypropyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-cyclopropyl-9-[(3-hydroxyphenyl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
7-(1-benzothiophen-3-yl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-ethyl-6-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
(2S,4R)-4-amino-1-(3-methanesulfonylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(4-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]-1,3-benzoxazole-6-carboxamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-6-methylpyrimidin-4-amine
1-{2-[4-(4-chlorophenyl)butanamido]ethyl}piperidine-3-carboxamide
1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazole
1-(3-fluorophenyl)-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
(1s,4s)-4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclohexan-1-ol
N-(oxolan-2-ylmethyl)-1-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}quinoline-5-carboxamide
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-methoxyacetyl)-N-methyl-N-(quinoxalin-2-ylmethyl)piperidine-4-carboxamide
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-(1-{1-[(4-methoxyphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
3-ethyl-5-{3-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]phenyl}-1,2,4-oxadiazole
(5-{[4-(4-chlorophenyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-benzyl-1-(1-cyclobutanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
(1S,5R)-3-[(2,3-difluoro-4-methylphenyl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)propyl]-2,3-dihydro-1H-isoindole
(4aR,7aS)-1-butanoyl-4-(3-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-{5-[1-(furan-3-ylmethyl)pyrrolidin-2-yl]thiophene-2-carbonyl}thiomorpholine
1-[4-({4-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(3-methoxypropyl)piperidine
3,5-dimethyl-1-{4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
3-ethyl-1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
(2R,6R)-4-[(3-hydroxy-4-methoxyphenyl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol