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3-(4-methoxyphenyl)-3-phenyl-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
methyl 7-oxo-9-(pyridin-3-ylmethoxy)-3-{spiro[2.4]heptane-1-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[4-(dimethylamino)naphthalene-1-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propylsulfanyl)ethan-1-one
2,3-dimethoxy-N-({1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}methyl)benzamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-(dimethylsulfamoyl)-5-[(furan-3-ylmethyl)amino]benzamide
N-[(3R,4S)-1-[5-(piperidine-1-carbonyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
5-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-propylpyrimidine-5-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-3-yl)quinoline-4-carboxamide
4-methyl-6-[2-(3-phenylpropyl)morpholine-4-carbonyl]pyrimidin-2-amine
4-[(4-fluorophenyl)methyl]-1-(2-methyl-1,3-thiazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-N-ethylpyrimidin-4-amine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-6-methoxypyrimidin-4-amine
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-phenylbutan-1-one
N-(2-ethylphenyl)-3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1S,4S)-5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
6-[(E)-2-cyclohexylethenyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
2-ethyl-9-(6-methoxypyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,3-dihydroxypropan-2-yl)acetamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
[4-benzyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-yl]methanol
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-[2-(phenylsulfanyl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
8-(3-hydroxybenzoyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N-methyl-6-oxo-1-(pyridin-2-ylmethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-3-carboxamide
2-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}quinolin-4-ol
(4aS,7aR)-1-cycloheptanecarbonyl-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-methanesulfonamido-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
3-(1H-imidazol-2-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]benzamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-ol
2-[4-(4-cyclohexylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
{1-[1-(4-methoxy-3,5-dimethylbenzoyl)piperidin-3-yl]piperidin-4-yl}methanol
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine
2-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}benzoic acid
N-(1-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-1H-pyrazol-5-yl)acetamide
1-(1H-imidazole-4-carbonyl)-3-(4-phenylbenzoyl)piperidine
1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}piperidin-3-ol
(3S,4S)-1-(1H-indol-4-ylmethyl)-4-(3-methoxyphenyl)piperidin-3-ol
(1-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-4-methylpiperazin-2-yl)methanol
4-(3,6-dimethylpyrazin-2-yl)-2-{[(2-methoxyethyl)amino]methyl}phenol
N,N-dimethyl-4-oxo-4-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}butanamide
(3S,9aR)-8-(4-fluorobenzoyl)-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one