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2-(2,6-dimethylpyrimidine-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-chloro-N-[2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2,2-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
2-[1-methyl-5-(thiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
{9-[(3-fluorophenyl)methyl]-3-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
8-(5-ethylthiophene-3-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-benzyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-5-formamido-1-methyl-1H-1,3-benzodiazole-7-carboxamide
1-[benzyl(methyl)amino]-3-(5-{[(cyclohexylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyridine-4-carbonitrile
4-[4-(carbamoylmethyl)phenyl]-2-chlorobenzamide
N-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-chlorobenzamide
(3aR,6aR)-2-[(4-chloro-2-fluorophenyl)methyl]-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-N,N-diethyl-2-oxoacetamide
2-{[2-methyl-2-(methylcarbamoyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-[3-(1H-imidazol-1-yl)propyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
7-(oxan-4-yl)-N-[2-(pyridin-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(1H-indol-1-yl)ethyl]propanamide
5-[(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)sulfonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,3-oxazole-5-carboxamide
5-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
3-(2-hydroxyphenyl)-N-{2-[methyl(phenyl)amino]propyl}-1H-pyrazole-5-carboxamide
2-(3-chloro-4-hydroxyphenyl)-N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)acetamide
4-acetyl-N-(1H-1,2,3-benzotriazol-4-yl)-1,4-diazepane-1-carboxamide
N,N-dimethyl-6-[2-(1,3-thiazol-2-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(cyclopropylmethyl)({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-[4-(1-hydroxypropyl)piperidin-1-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-4-(thiophen-2-yl)butan-1-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,3-thiazole-5-carboxamide
5-(1-benzylpiperidin-4-yl)-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
1-[(4-fluorophenyl)methyl]-1-(3-hydroxypropyl)-3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
9-{2-[ethyl(methyl)amino]butanoyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(1-methylpiperidin-3-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[1-(1-benzofuran-5-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
4-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
1-(2,2-dimethylpropyl)-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-ol
7-(3-chlorophenyl)-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
5-amino-4-chloro-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-cyclooctyl-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
1-[2-methoxy-5-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-(5-methyl-1,2-oxazol-3-yl)-2-(2-methylbutanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}phenol
[3-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}methyl)-2,4,6-trimethylphenyl]methanol
{1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
2-{4-[(2-cyanophenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
(2S)-2-[4-(4-acetylphenyl)piperazine-1-carbonyl]pyrrolidine-1-carboxamide