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1-[2-(propylsulfanyl)phenyl]-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
1-ethyl-4-{[methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
1-[(3,5-dimethylphenyl)methyl]-4-(2-methylpyridin-4-yl)piperazin-2-one
(3aS,6aS)-2-[(3-ethenylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl (2S,4S)-4-acetamido-1-[(4-methylphenyl)methyl]pyrrolidine-2-carboxylate
{1-cycloheptanecarbonyl-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2,1-benzoxazole-3-carboxamide
3-fluoro-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
{1-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}(methyl)(pyridin-2-ylmethyl)amine
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-4-fluoro-3-hydroxybenzamide
3,7-dimethyl-11-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3,7,11-triazaspiro[5.6]dodecane
2-(4-fluorophenyl)-N-[1-(pyridin-3-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
3-phenyl-5-(thiophene-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-cyclopentyl-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(5-ethylpyridin-2-yl)methyl]piperidine-4-carboxylic acid
N-(2,4-difluorophenyl)-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)benzamide
3-(1H-imidazol-2-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(2-oxooxolan-3-yl)propanamide
3-(furan-2-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
2-[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
N-[3-(5-methyl-4-{[2-(1,3-thiazol-4-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]-3-(pyridin-3-yl)propanamide
6-(2,2-diphenylpropyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-cyclohexyl-4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
(3S,9aR)-3-methyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[(1,4-dioxan-2-ylmethyl)amino]methyl}-6-fluoroquinolin-4-ol
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyridin-3-yloxy)ethan-1-one
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-4-(morpholin-4-yl)benzamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
(2S,4S)-4-amino-N-methyl-1-[(4-methylphenyl)methanesulfonyl]pyrrolidine-2-carboxamide
2-(2-cyclopropylpyrimidin-5-yl)-4-(3,3-dimethylpyrrolidine-1-carbonyl)-6-fluoroquinoline
N-methyl-N-[(5-methylfuran-2-yl)methyl]-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
1-phenyl-4-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,4-diazepane
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(1,2,2-trimethylpyrrolidin-3-yl)methyl]amine
N-ethyl-1-methyl-3-(propan-2-yl)-N-(2,2,2-trifluoroethyl)-1H-pyrazole-5-carboxamide
5-(methoxymethyl)-N-[4-(5-methyl-4-{[(1-methylcyclohexyl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-[3-oxo-3-(3-phenylpiperidin-1-yl)propyl]pyrrolidin-2-one
5-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(3S)-3-benzyl-4-{[3-(2-hydroxyethoxy)phenyl]methyl}piperazin-2-one
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-benzyl-N-[(3-methylpyridin-2-yl)methyl]-3-(2-oxopiperidin-1-yl)propanamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
9-(2-methoxyethyl)-1-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-4-hydroxy-2-[(phenylsulfanyl)methyl]-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide