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1-[(3-methylphenyl)methyl]-4-[2-(pyridin-2-ylsulfanyl)propanoyl]piperazin-2-one
5-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-1-azabicyclo[3.2.1]octane
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-methylpentane-1,2-dione
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
1-[(3-fluorophenyl)methyl]-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
(3S,9aR)-3-methyl-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-butyl-1H-imidazol-4-yl)-1-(pyrrolidin-3-yl)-1H-imidazole
N-{2-[3-(aminomethyl)pyrrolidin-1-yl]-2-oxoethyl}-4-ethylcyclohexane-1-carboxamide
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-({3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
1-[(4-fluorophenyl)methyl]-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
8-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-ethyl-4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}morpholine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-5-methoxy-N-(propan-2-yl)benzamide
2-{[4-(3-cyano-4,6-dimethylpyridin-2-yl)piperazin-1-yl]methyl}benzoic acid
1-{4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
1-(furan-2-ylmethyl)-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
[(1-cyclopentylpiperidin-4-yl)methyl][(2-fluoro-5-methoxyphenyl)methyl](oxolan-2-ylmethyl)amine
4-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyrimidin-2-amine
5-{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
4-{[2-(1-cyclobutanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
2-[1-(2,2-dimethylpropyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(3-cyano-4-methoxyphenyl)-3-[(1-methanesulfonylpiperidin-3-yl)methyl]urea
3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
3-(4-chlorophenyl)-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
3-{5-[(3-hydroxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
2,2-dimethyl-N-(1-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
methyl (2S,4R)-4-[2-(4-fluorophenyl)acetamido]-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxylate
N-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-[3-(5-chlorothiophen-2-yl)-4-methoxyphenyl]ethan-1-amine
N-{4-oxo-4-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butyl}acetamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
6-(4-methylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
6-(2-methoxyphenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyridazin-3-amine
(3S,4R)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
1-(2-fluorophenyl)-4-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}piperazine
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-[(diethylamino)methyl]-5-ethyl-N-(2-methylprop-2-en-1-yl)furan-2-carboxamide
N,N-dimethyl-5-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}pyridin-2-amine
1-ethyl-3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
1-[(2-chlorophenyl)methyl]-N-(3-hydroxy-2,2-dimethylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-[1-(2-methylpropyl)-4-(1H-pyrazole-4-carbonyl)piperazin-2-yl]ethan-1-ol
1-benzyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-(4-phenylbutyl)oxane-2-carboxamide
N-{[8-(1H-1,3-benzodiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
ethyl 1-ethyl-5-(1-methylpiperidine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate