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4-(2,6-dimethylpyridin-3-yl)-2-(1H-pyrazol-3-yl)pyrimidine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidin-3-yl]acetamide
(3S,4S)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-({[(3R,4R)-1-(2,3-dimethylquinoxaline-6-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
methyl 5-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)thiophene-2-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
8-{5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl}quinoline
(4aR,7aS)-1-methyl-4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
4-methyl-6-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-benzothiazol-2-amine
2-[2-(4-fluorophenyl)piperidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
4-[(2-ethoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(3-chloropyridin-2-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
[4-(3-phenylpropyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-yl]methanol
[2-methoxy-1-(pyridin-2-yl)ethyl][(2-methoxy-3,5-dimethylphenyl)methyl]methylamine
4-hydroxy-2-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinoline-6-carboxamide
8-(2-ethoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(2-chloro-4-fluorophenyl)methyl]-3-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}piperazin-2-one
3-(2,3-dihydro-1,4-benzodioxin-2-ylformamido)-N-(2-methylphenyl)propanamide
5-(4-methylpiperidine-1-carbonyl)-4-oxo-N-[(4-phenyloxan-4-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-[4-(2-phenylethyl)piperidine-1-carbonyl]piperidin-2-one
3-hexyl-8-[2-(2-oxopyrrolidin-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)morpholine
2-[4-(isoquinolin-5-ylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
6-ethyl-2-(piperidin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrimidin-4-amine
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-3-[3-(pyrrolidin-1-yl)propyl]-1,2,4-oxadiazole
N-methyl-N-(1-methylpiperidin-4-yl)-3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
4-(1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)morpholine
1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-[(3R)-pyrrolidin-3-yl]urea
(4aS,7aR)-1-(2,5-dimethylbenzoyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2S,4S)-4-(5-chlorothiophene-2-amido)-1-methylpyrrolidine-2-carboxylate
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(2,5-dimethoxyphenyl)pyrrolidine
5-[3-(3-benzoylpiperidin-1-yl)-3-oxopropyl]-5-benzylpyrrolidin-2-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]oxy}benzamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-[4-(pyrrolidin-1-yl)butyl]piperidine-3-carboxamide
4-(cyclopropylamino)-5-methyl-N-[phenyl(pyridin-4-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-methylfuran-3-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(3S,4R)-1-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
3-[(3R,4R)-4-amino-3-hydroxypiperidine-1-carbonyl]-8-methyl-1,4-dihydroquinolin-4-one
3-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
1-[(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
(1S,6R)-9-[3-(methoxymethyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
(3aR,6aR)-2-acetyl-5-({[2-(4-fluorophenyl)ethyl]carbamoyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-phenoxyethyl)-2-(propan-2-yl)-1H-imidazole
dimethyl(3-{2-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}thiomorpholine
(3S,4R)-1-(2H-1,3-benzodioxol-4-ylmethyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol