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1-(4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)urea
N,N-dimethyl-2-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-sulfonamide
3-(2-methylphenyl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-8-azabicyclo[3.2.1]octane
(2S)-N-[(3-methoxyphenyl)methyl]-2-phenyl-N-(prop-2-en-1-yl)butanamide
3-[({2-[2-(trifluoromethoxy)phenyl]ethyl}amino)methyl]pyrrolidin-3-ol
3-{1-[(4-methoxypiperidin-1-yl)sulfonyl]piperidin-3-yl}benzoic acid
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-4-(pyridin-4-yl)pyrimidin-2-amine
2-(2-aminoethyl)-5,6-dimethyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]thieno[2,3-d]pyrimidin-4-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(pyridin-3-yl)propanamide
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
4-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-amino-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-(3,4-dimethylphenyl)-1-(4-fluorobenzoyl)piperidin-3-amine
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carbonyl)morpholine
(3S,4S)-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-4-methylpiperidine-3,4-diol
2-fluoro-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-sulfamoylbenzamide
(3-{2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1,3-dimethyl-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-one
3-(1H-imidazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}butanamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-benzyl-4-(furan-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-tert-butyl-N-(cyclohexylmethyl)-4-hydroxypyrimidine-5-carboxamide
1-{5-[3-(5-methylfuran-2-yl)butyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-ol
N-(furan-2-ylmethyl)-2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
6-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamine
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-ethylbutan-1-one
N-[3-(furan-2-yl)phenyl]-1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidine-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl][(8-methoxyquinolin-2-yl)methyl]methylamine
N-(1-{[3,5-dichloro-4-(propan-2-yloxy)phenyl]methyl}pyrrolidin-3-yl)acetamide
2-(cyclopropylmethyl)-9-(1H-1,2,4-triazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-(furan-2-amido)-5-{[1-(2-methoxyphenyl)propan-2-yl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
N-ethyl-7-[(3-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N,3-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(2-phenoxyethyl)piperazine
1-(2,6-difluoro-3-methoxybenzoyl)-2-(3-methoxypropyl)piperidine
3-{2-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-4,6-dimethyl-2,3-dihydro-1H-indol-2-one
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
2-(4H-1,2,4-triazol-4-ylmethyl)-3,4-dihydroquinazolin-4-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
3-(4-methoxypyrimidin-2-yl)benzonitrile
N-(2-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
(2S,3R)-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methyl-2-(methylamino)pentan-1-one