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2-(pyridin-2-ylmethyl)-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
(2S,4R)-N,N-diethyl-4-(3-hydroxybenzamido)-1-(3-hydroxypropanoyl)pyrrolidine-2-carboxamide
(4S)-1-(3-chloro-5-methoxybenzoyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(2-methoxyethyl)piperidine
4-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2,1,3-benzoxadiazole
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
N-[2-(dimethylamino)ethyl]-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(3-phenyl-1,2,4-oxadiazol-5-yl)-4-(piperidine-1-carbonyl)piperidine
(3aR,6aR)-2-acetyl-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}morpholin-3-yl)acetic acid
2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-1,3-benzodiazole-6-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-[1-(1,3-dihydroxypropan-2-yl)piperidin-3-yl]propan-1-one
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
(1S,2S,3R,4R)-3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]bicyclo[2.2.1]heptan-2-amine
(2S,4R)-1-benzyl-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-methylpyrrolidine-2-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(3-methylphenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[3-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-5-methyl-1,2-oxazol-4-yl]methanol
5-[3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-oxopropyl]-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
ethyl 1-(2,3-dimethylphenyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-1H-pyrazole-4-carboxylate
N-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}cyclohexanamine
3-[(3-methoxyphenyl)methyl]-8-(2-methylbutyl)-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-{4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
4-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
6-methoxy-3-methyl-N-(2-oxoazepan-3-yl)-1-benzofuran-2-carboxamide
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3,4-dimethylbenzamide
3-(1,5-dimethyl-1H-indazole-3-carbonyl)-3,9-diazaspiro[5.5]undecane
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,5-dioxo-1-propylimidazolidin-4-yl)acetamide
2-(dimethylamino)-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[(2R,3R)-2-hydroxy-1'-[(1-methyl-1H-indol-3-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-(2-methoxyethyl)-2-(2-oxopiperidin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
N-({7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
1-[(1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-fluoro-N-methyl-4-(morpholin-4-yl)pyrimidin-2-amine
1-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)naphthalene-2-sulfonamide
(1S,3R)-3-amino-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}cyclopentane-1-carboxamide
1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazole
(4aR,7aS)-1-benzyl-4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
4-benzyl-3-ethyl-1-(5-fluoro-2-methoxybenzoyl)-1,4-diazepan-5-one
methyl 7-oxo-3-[(4-oxo-4H-chromen-3-yl)methyl]-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(3-chlorophenyl)ethyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-aminoethyl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]quinazolin-4-amine