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7-(3-chlorophenyl)-4-propyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{5-[3-(4-methylpiperazin-1-yl)butyl]-1,2,4-oxadiazol-3-yl}pyridazine
{[2-(cyclopentyloxy)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
1-{7-[(2R)-oxolane-2-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-ol
(1S,4S)-2-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
1-ethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
3-{5-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
methyl 2-[butyl(methyl)sulfamoyl]-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-[2-(pyrrolidin-1-yl)ethyl]benzene-1-sulfonamide
(3aS,6aS)-5-cyclopentanecarbonyl-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[ethyl(pyridin-4-ylmethyl)amino]-N-(2-methoxy-5-methylphenyl)piperidine-1-carboxamide
N-(4-chloro-3-methoxyphenyl)-2-{[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}acetamide
N-[(3R,4S)-1-(3-hydroxypropyl)-4-phenylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-(2-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(adamantan-1-yl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(oxan-4-yl)-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
3-methyl-5-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]pyrrolidin-3-yl]methanol
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-indazole-3-carboxamide
2-({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}(methyl)amino)acetamide
1-ethyl-3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
N-methyl-N-(1,3-thiazol-2-ylmethyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
4-(pyrrolidin-1-ylmethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}benzamide
1-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-phenylpiperazine
2-{[4-(2,2-dimethoxyethyl)piperazin-1-yl]methyl}quinoline
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methoxyphenyl)methyl]-2-(morpholin-3-yl)acetamide
2-{1-methyl-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
4-acetamido-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)-1-methyl-1H-1,3-benzodiazole
methyl (4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
5-(1-methylcyclopropanecarbonyl)-3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(3-chlorophenyl)-4-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}piperazine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-4-methyl-2-oxopentanamide
N-[(2-chlorophenyl)methyl]-3-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)propanamide
(2S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidine-2-carboxamide
N-[4-(2-methoxyphenoxy)phenyl]-2-propylpyrrolidine-1-carboxamide
5-(naphthalen-1-yl)-N-(oxan-4-ylmethyl)-1,2,4-triazin-3-amine
2-(2-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
1-(naphthalen-1-ylmethyl)-N-[(3S)-2-oxoazepan-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]-N-phenylpropanamide
3-(3-chlorophenyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-3-phenylpropanamide
(2S)-2-amino-N-butyl-N-(thiophen-3-ylmethyl)propanamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}urea
2,3,6-trimethyl-4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
1-{6-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-2-yl}ethan-1-ol
(3S,4S)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid