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N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
N-[2-(4-cyclopentylmorpholin-2-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
6-methoxy-3-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1-benzofuran-2-carboxamide
(4aS,7aR)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
3-(3-fluorophenyl)-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}prop-2-ene-1-sulfonamide
5-(5-methyl-1,3-oxazol-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
(1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperidin-3-yl)methanol
2,8-dimethyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)quinoline-4-carboxamide
1-[4-(azepan-1-ylmethyl)phenoxy]-3-[benzyl(methyl)amino]propan-2-ol
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-3-(2-hydroxyethyl)piperazin-2-one
1-[2-(2-chlorophenyl)ethyl]-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
(1R,3S)-3-amino-N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methylcyclohexane-1-carboxamide
4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
3-chloro-N-[(3R,4S)-1-[2-(methylcarbamoyl)ethyl]-4-propylpyrrolidin-3-yl]thiophene-2-carboxamide
(1r,4r)-4-({[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}methyl)cyclohexane-1-carboxamide
ethyl 2-(1-{1-[(2-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
6-[(diethylamino)methyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{[3-(difluoromethoxy)phenyl]methyl}-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
(3aR,7aS)-N-(dimethyl-1,2-oxazol-4-yl)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
1-cyclopentyl-N3-(3-methylbutyl)-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine
2-(2H-1,2,3-benzotriazol-2-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(4-methoxybenzoyl)piperidine-3-carboxylate
ethyl 4-{4-[5-(3-methylbutanamido)-1H-pyrazol-1-yl]piperidin-1-yl}piperidine-1-carboxylate
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-(1H-imidazol-2-yl)benzamide
4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine
7-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2-oxa-7-azaspiro[4.5]decane
5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]urea
2-[4-(1-phenylpiperidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
4-ethyl-3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(dimethylamino)ethyl]-2-acetamido-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)acetamide
2-(2-methoxyethyl)-N-[2-methyl-3-(3-methylbutanamido)phenyl]piperidine-1-carboxamide
N-cyclopentyl-2-[4-(6-oxo-3-phenyl-1,6-dihydropyridazin-4-yl)piperazin-1-yl]propanamide
1-ethyl-8-(1H-indol-2-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(2-methoxyphenyl)methyl]-N-methylpiperidin-3-amine
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
2-amino-4-[5-(oxan-2-yl)thiophen-2-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
4-({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)-1,4-diazepane-1-carbaldehyde
1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
ethyl 2-(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)acetate
[5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
1-[(1-methylpiperidin-2-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-benzyl-3-({1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}oxy)benzamide