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7-[(2-methoxy-4-methylphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{3-[(3-methoxyphenyl)methyl]-1-[4-(morpholin-4-yl)benzoyl]piperidin-3-yl}methanol
(2R,6R)-1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
(2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylamino)propanamide
N-{1-benzyl-7-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-2-methyl-1H-1,3-benzodiazol-5-yl}acetamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(3-methylthiophene-2-carbonyl)piperidine-3-carboxylate
2-[(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]acetic acid
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]azepan-4-ol
3-(4-methyl-1,3-thiazol-5-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
N-(4-chloro-2-fluorophenyl)-2-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}acetamide
3-({1-[1-(thiophen-2-yl)propyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-(2-methoxy-4-methylphenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-(oxan-4-yl)piperidine-3-carboxamide
4-({5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
methyl 5-{[(3,4-dimethylphenyl)methyl]amino}-3-acetamido-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[3-(azepan-1-yl)-2-hydroxypropyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[5-({cyclopropyl[(3-methylthiophen-2-yl)methyl]carbamoyl}amino)-2-fluorophenyl]acetamide
2-amino-4-[5-(oxan-2-yl)furan-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(1,3-benzothiazol-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
3-(2-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-phenoxypropanamide
2-(4-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrazine
2-{2-oxo-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-1-yl}benzonitrile
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
5-{2-[3-(2-fluorophenoxy)azetidine-1-carbonyl]phenyl}-1H-1,2,3,4-tetrazole
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
2-(2-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenoxy)acetic acid
1-[(3-chlorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-(3-acetylphenoxymethyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-butyl-5-(4-methoxypiperidine-1-carbonyl)-1,3-benzoxazole
2-methyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
methyl 3-[({5-methyl-2-[3-(2-methylfuran-3-amido)phenyl]-1,3-oxazol-4-yl}methyl)carbamoyl]benzoate
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(morpholin-4-yl)ethyl]acetamide
methyl 2-hydroxy-5-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]benzoate
1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-methoxy-2-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-(5-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)benzonitrile
5-{1-[(benzylsulfamoyl)amino]ethyl}-1,3,4-thiadiazol-2-amine
1-[3-(2,4-dimethoxyphenyl)-4-(morpholin-4-yl)phenyl]ethan-1-one
{[2-(furan-2-yl)phenyl]methyl}(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
(1S,5R)-3-(3-methyl-1H-pyrazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-({2-[2-(cyclopropylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
5-[4-(dimethylamino)piperidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(diphenylmethyl)-N-[2-(2-methylphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-butyl-4'-[2-(ethylsulfanyl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one