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8-[2-(methylsulfanyl)pyrimidin-4-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{5-[(diethylamino)methyl]-2-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
(2S,4R)-N-cyclopropyl-4-[(4-fluorophenyl)sulfanyl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-(2-methoxyethyl)-N-methyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(1-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
[1-(oxan-4-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
(1R,5R)-6-(2,6-dichlorobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(5S,9aS,9bS)-5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-({[2-(4-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
[(3S,4S)-4-(hydroxymethyl)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
(3R,4S)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-propylpyrrolidin-3-amine
1-(2-ethoxyethyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-1H-pyrazole-5-carboxamide
2-cyclohexyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
5-ethyl-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}thiophene-2-carboxylic acid
2-(morpholin-4-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-(pyridin-3-yl)acetamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})[3-(morpholin-4-yl)propyl]amine
1-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholin-4-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
methyl 7-oxo-3-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-8-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2-ethyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-(2-{8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)acetamide
{[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-{[7-(3-chloro-2-fluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N,N-diethyl-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-amine
dimethyl[(6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]amine
1-(4-methylpiperazin-1-yl)-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]propan-1-one
1-cyclopentyl-3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-(4-{4-[(naphthalen-1-ylmethyl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]morpholin-4-yl}butan-1-one
N-[(2R,3R)-1'-(2-cyclopentylacetyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
N-[2-(2-methylpropanesulfonyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-(1H-pyrazol-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-fluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-1-butyl-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(2S,4R)-4-[(1-benzylpiperidin-4-yl)amino]-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2-methoxyphenyl)methyl]-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetamide
3-hydroxy-N-[(3R,5S)-1-(oxan-4-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]pyridine-2-carboxamide
2-(2-methoxyphenoxy)-2-methyl-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}propan-1-one
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-[(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]morpholine
N-({1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl}methyl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-methyl-1,3-thiazole-4-carboxamide
N-(pyridin-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-oxopiperidin-1-yl)-N,N-bis(pyridin-3-ylmethyl)acetamide
N-benzyl{[4-(1H-1,2,4-triazol-1-yl)phenyl]amino}sulfonamide