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5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
N-(1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
4-[(dimethylamino)methyl]-1-(2-ethylpyrimidine-5-carbonyl)azepan-4-ol
2-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-thiazole-4-carboxamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2-dimethylpropan-1-one
[1-(2-fluorobenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
4-{1-methyl-4-[4-(pyrrolidin-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-[1-(7-fluoro-4,6-dimethylquinazolin-2-yl)piperidin-4-yl]-4-(pyridin-2-yl)piperidin-4-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 4-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)benzoate
1-(pyrrolidin-3-yl)-4-{[2-(trifluoromethoxy)phenyl]methyl}piperazine
1-(2-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
1-[3-(furan-2-yl)-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
3-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}benzonitrile
1-(4-methoxyphenyl)-3-methyl-4-[(3-methyl-1-benzofuran-2-yl)methyl]piperazin-2-one
4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-oxazolidin-2-one
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[(4-chlorophenyl)methyl]-4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
N-[(2-chloro-4-fluorophenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(1S,4S)-2-(4-chloro-2-methoxy-5-methylphenyl)-5-(quinoline-2-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(3-cyclopentylpropyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
ethyl 4,4,4-trifluoro-3-[4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamido]butanoate
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-3-carboxamide
(1R,5S)-6-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}(pyridin-3-ylmethyl)amino)butan-1-ol
2-methyl-6-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-phenylbenzamide
1-{2-[(1-benzylpiperidin-4-yl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-(6-hydroxy-4-{thieno[3,2-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)acetic acid
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]propanamide
1-(3-methylpyridin-4-yl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
3-({1-[4-(morpholin-4-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
methyl 3-[3-(3,5-dimethylphenyl)propanoyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S)-1-[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carbonyl]pyrrolidine-2-carboxamide
N-(1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)methanesulfonamide
N-[3-(4-fluorophenyl)propyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-({1-[(2E)-4-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(1-{7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
{1-[(2,4-dimethoxyphenyl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
(3S,4S)-1-[(3-fluorophenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
[(3S,5R)-5-[(dimethylamino)methyl]-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperidin-3-yl]methanol
N-({5-[(2-phenoxyethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)acetamide
2-amino-6-(furan-2-yl)-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(1S)-1-[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine