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2-methoxyethyl 9-[(2-cyanophenyl)methyl]-3,9-diazaspiro[5.5]undecane-3-carboxylate
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-1,3-benzothiazole
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-4-phenylbutane-1,4-dione
methyl 4-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzoate
2,4-dimethoxy-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(1,4-oxazepane-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{1-[1-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N,N-dimethyl-4-[2-(4-methylpentyl)morpholin-4-yl]-4-oxobutanamide
3-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}imidazo[1,2-a]pyridine-2-carboxamide
methyl 2-{[(4-chlorophenyl)methyl]sulfamoyl}-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(pyrimidin-2-yl)pyrrolidin-3-yl]acetamide
N-cyclooctyl-1-(2-methoxyethyl)-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]benzamide
(3aR,5S,6S,7aS)-2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-octahydro-1H-isoindole-5,6-diol
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[(1-phenylcyclohexyl)methyl]acetamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(2-oxopiperidin-1-yl)butanamide
4-propyl-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-1,2,3-thiadiazole-5-carboxamide
4-({2-[(methylcarbamoyl)methyl]-3-oxopiperazin-1-yl}methyl)-N-(pyridin-3-yl)benzamide
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-6-[2-(propan-2-yloxy)phenyl]pyridazine
N-cyclopropyl-2-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}benzamide
1-[2-(2-methoxy-2-methylpropyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-3-carboxamide
N-cyclopropyl-1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
8-[(2-hydroxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethyl-1,2-oxazol-4-yl)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazole
6-methyl-5-{5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
N-methyl-2-(methylsulfanyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
9-{2-[2-(butan-2-yl)phenoxy]acetyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
7-({[(4-fluorophenyl)methyl](1-hydroxybutan-2-yl)amino}methyl)-4-methyl-2H-chromen-2-one
1-cyclopentyl-4-{2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetyl}piperazin-2-one
[(4-methanesulfonylphenyl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
1-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pent-4-en-1-one
1-(furan-2-ylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
methyl 2-(azocane-1-sulfonyl)-6-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}azepane-2-carboxamide
3-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl}benzoic acid
(3E)-2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-5,5-dimethylhex-3-enoic acid
1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxylic acid
1-{imidazo[1,2-b]pyridazin-6-yl}-4-(pyridin-4-ylmethyl)piperazine
1-(1-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}ethyl)-4-methylpiperazine
2-(3-chlorobenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
2-butyl-5-(2-methyl-4-phenylpiperazine-1-carbonyl)-1,3-benzoxazole
(1S,9S)-11-{2-[(prop-2-en-1-yl)amino]benzoyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-benzyl-8-[(3-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3,5-dimethyl-4-(5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)-1,2-oxazole