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ethyl[(1-methyl-1H-imidazol-2-yl)methyl]{[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
4-{[5-(1-cyclohexylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
N-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]methanesulfonamide
3-(1-ethyl-1H-imidazol-2-yl)-1-[1-(oxan-4-yl)piperidine-4-carbonyl]piperidine
3-(2-fluoro-3-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
3-(1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-3-yl)benzoic acid
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-amine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)-N-methylbenzamide
(1R,5S,6S)-6-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
3-[2-(4-fluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
2-[1-(1-cyclobutanecarbonylpiperidin-4-yl)-N-methylformamido]-2-(pyridin-3-yl)acetic acid
(2S)-2-(hydroxymethyl)-N-[3-(3-methoxyphenyl)phenyl]pyrrolidine-1-carboxamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-{4-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-(butan-2-yl)-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
2-(1-benzyl-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
1-[(2-methylphenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-({[(3R,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
5-ethyl-2,3-dimethyl-N-[2-(4-methylpiperazin-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
2-amino-4-({[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}amino)quinazoline-6-carboxylic acid
(2R)-2-amino-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-phenylacetamide
1-(1H-imidazol-2-ylmethyl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
N-(2-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)carbamoyl]amino}ethyl)pyridine-3-carboxamide
2-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-(3-methylpiperidin-1-yl)-3-{[(5-phenyl-1H-pyrazol-3-yl)methyl]amino}propan-1-one
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(methylsulfanyl)acetamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[1-(4-fluorophenyl)piperidin-4-yl]propanamide
N-butyl-N-methyl-3-({[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(2-methoxyphenyl)-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(3-phenylpyrrolidin-1-yl)ethan-1-one
ethyl 2-[(4-acetyl-1,4-diazepan-1-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methanol
4-(3-{4-[1-(dimethylamino)ethyl]piperidine-1-carbonyl}phenyl)phenol
4-{4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[2-(furan-2-yl)ethyl]piperidin-4-amine
1-[(3-fluoro-2-methylphenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(2S,4S)-4-amino-N-methyl-1-{2-methyl-3-[(pyridin-2-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
[(2S)-1-{[1-(1-cyclopentylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}pyrrolidin-2-yl]methanol
1-({1-[(4-methylphenyl)carbamoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
6-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
3-{[1-(2-phenylacetyl)pyrrolidin-3-yl]methyl}benzoic acid
1-{3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
3-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-6-(morpholin-4-yl)pyrimidin-2-amine