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3-({1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
1-[4-(thiomorpholine-4-carbonyl)phenyl]pyrrolidin-2-one
(5S,9aS,9bS)-2-methyl-5-[4-(5-methylfuran-2-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[(cycloheptylamino)methyl]-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
5-fluoro-2-(1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
3-[(3R,4S)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-N-methylpiperidine-2-carboxamide
N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1H-indol-4-ylmethyl)-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
3-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-2-(methylsulfanyl)pyridine
N-cyclopropyl-5-(1H-indazole-3-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[4-(1,2-oxazol-3-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-(4-{[(1S)-1-phenylethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
1-[2-(1-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
3-(azetidine-1-carbonyl)-N-[(5-methylpyrazin-2-yl)methyl]benzene-1-sulfonamide
2-(2-chlorophenyl)-N-(1,3-dihydroxypropan-2-yl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
[(4-{[1-(2,5-dimethoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-[2-(dimethylamino)-1-phenylethyl]-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-cyclobutyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}propan-1-one
2,6-dimethyl-4-[({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amino)methyl]phenyl acetate
(2E)-1-[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(thiophen-2-yl)prop-2-en-1-one
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypyrazine
4-[4-(cyclopentylmethyl)piperazin-1-yl]-5,6-dimethylpyrimidine
[4-(5-methylpyrazine-2-carbonyl)-1,4-oxazepan-6-yl]methanol
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(pyridin-3-yl)piperazine
2-cyclopropyl-N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-4-methylpyrimidine-5-carboxamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-4-(trifluoromethyl)pyrimidin-2-amine
1-(2-methoxyphenyl)-5-(5-methyl-1,2-oxazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
5-{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2-(pyridin-3-yl)morpholine
(2S,4S)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(pyridin-2-ylsulfanyl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
(1-{[5-(3,4-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}cyclobutyl)methanol
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N,6-dimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-propylpyrimidin-4-amine
[(5-fluoro-1H-indol-2-yl)methyl]({[2-(methoxymethyl)pyrimidin-5-yl]methyl})methylamine