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4-(2,4-dimethylpyrimidine-5-carbonyl)-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
4-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
ethyl 2-[1-(5-chloro-2-fluorobenzoyl)piperidin-2-yl]acetate
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]thiophene-3-carboxamide
1-(naphthalene-1-sulfonyl)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
8-(1-hydroxypropan-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2-azaspiro[4.5]decan-3-one
(2R)-2-amino-3-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(4-methyl-2-phenyl-1H-imidazol-1-yl)acetamide
methyl 9-[3-(dimethylamino)propoxy]-7-oxo-3-[2-(piperidin-1-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methyl-5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
4-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methoxyphenol
1-(4-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}piperidin-1-yl)ethan-1-one
N-[(3S,4R)-1-(3-fluoropyridin-4-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
6-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2,3-dimethylquinoxaline
1-ethyl-4-{[3-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
(1s,4s)-4-[2-(8-chloroquinolin-2-yl)-1H-imidazol-1-yl]cyclohexan-1-amine
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
N-[(2R,3R)-1'-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-3-yl]methanol
1-(1,4-dithiepan-6-yl)-3-(pyrrolidin-1-yl)piperidine
1-methyl-N-[(6-methylpyridin-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-(2-fluorophenoxymethyl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1,3-oxazole-4-carboxamide
6-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)pyrimidin-4-ol
2-[(1S,5R)-3-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-[2-(butan-2-yl)phenoxy]-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}acetamide
6-{3-oxo-3-[3-(4-phenylbenzoyl)piperidin-1-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
N,N-diethyl-1-[(1s,4s)-4-(5-chlorothiophene-2-sulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
(3S,4S)-3-hydroxy-4-[(2-methylquinolin-4-yl)amino]-1λ6-thiolane-1,1-dione
(1r,4r)-4-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}cyclohexan-1-ol
N4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N4-methyl-6-(pyrrolidin-1-yl)pyrimidine-2,4-diamine
4-[3-(benzyloxy)azetidine-1-carbonyl]-1-cyclopropanecarbonylpiperidine
5-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]isoquinoline
1-[(3-methoxyphenyl)methyl]-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-2-one
N-(2-methoxyethyl)-N-methyl-2-[1-(3-methylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N,15-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-9-(3-methylthiophen-2-yl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
4-[(dimethylamino)methyl]-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}azepan-4-ol
1-benzyl-6-(cyclopropylmethoxy)-4-(2,3-dihydro-1-benzofuran-2-carbonyl)-1,4-diazepan-2-one
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]benzonitrile
methyl 2-(1-{[(1H-1,3-benzodiazol-2-yl)carbamoyl]methyl}-3-oxopiperazin-2-yl)acetate
N-(1,3-benzothiazol-2-ylmethyl)-N,6-dimethyl-4-oxo-4H-pyran-2-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-(2,2-dimethylpent-4-en-1-yl)-2-methyl-1,4-diazepan-5-one