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2-[4-(methylsulfanyl)phenyl]-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]acetic acid
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(4-oxo-1,4-dihydropyridin-1-yl)acetamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1,2-oxazol-3-ylmethyl)acetamide
(1S,5R)-3-(3-phenylpropyl)-6-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{3-[cyclopentyl(methyl)amino]propyl}-2-(propan-2-yl)pyrimidine-5-carboxamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[2-(pyridin-2-yl)ethyl]-decahydro-2,7-naphthyridin-4a-ol
4-(cyclohexylmethyl)-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-5-ethyl-1,3-oxazole-4-carboxamide
(4aS,8aR)-6-[2-(1H-pyrazol-1-yl)acetyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[4-(benzyloxy)piperidin-1-yl]-2-(4-chloro-1H-pyrazol-1-yl)ethan-1-one
[(2-ethylpyrimidin-5-yl)methyl](methyl){[3-(trifluoromethyl)phenyl]methyl}amine
(3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-5-methyl-1,2-oxazol-4-yl)methanol
[5-({[2-(3,5-dimethylphenoxy)ethyl](methyl)amino}methyl)-2-methoxyphenyl]methanol
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-methyl-1-oxopropan-2-yl)thiophene-2-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
N,N-diethyl-3-methyl-4-{[(5-oxo-1-propylpyrrolidin-3-yl)carbamoyl]amino}benzamide
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
3-{1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[2-(4-methoxyphenyl)ethyl]-N-(oxolan-2-ylmethyl)-1H-imidazole-5-carboxamide
3-chloro-4-fluoro-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-benzothiophene-2-carboxamide
N2,N2-dimethyl-N4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
ethyl 1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
methyl 3-(2-methoxyacetamido)-5-{[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S)-2-amino-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]hexan-1-one
3-(1-{1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-1-ol
5-methanesulfonyl-4-(piperidin-3-yl)-2-[4-(propan-2-yl)piperazin-1-yl]pyrimidine
7-[(3-methylphenyl)methyl]-6-oxo-N-propyl-2,7-diazaspiro[4.5]decane-2-carboxamide
4-(6-phenylpyridazin-3-yl)piperazine-2-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]piperidin-3-yl]methanol
2-{1-[(2-ethoxyphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-2-one
4-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-1,4-diazepan-2-one
3-(3,4-dimethoxyphenyl)-N,N-dimethylpyrazin-2-amine
N-[(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(1H-pyrazol-1-yl)benzamide
1-[4-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)thiophen-2-yl]ethan-1-one
3-[(4aR,7aS)-4-methanesulfonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(2S,4S)-4-amino-N,N-diethyl-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidine-2-carboxamide
6-{[3-cyclopropyl-1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N,2,3,5-tetramethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
3-[3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]-1-methyl-1H-indole
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
ethyl 1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
8-[1-(3,4-difluorophenyl)piperidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
5,6-dimethyl-3-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one