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3-(azetidine-1-sulfonyl)-N-methyl-N-(oxan-2-ylmethyl)benzamide
5-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidine-1-carboxamide
2-[2-(ethylsulfanyl)ethyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-(morpholin-3-yl)acetamide
4-{2-methoxy-5-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}morpholine
3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-(naphthalen-2-yl)urea
2-{4-[3-(azepane-1-carbonyl)-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenol
1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-(methoxymethyl)pyrrolidine
5-benzenesulfonamido-1-ethyl-2-methyl-N-[1-(thiophen-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-(4-methoxyphenyl)propanamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(3-methoxypropanoyl)piperidine-4-carboxylate
5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,1-dimethylazepane-2-carboxamide
9-(but-3-yn-1-yloxy)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
(2S)-2-(methoxymethyl)-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)pyrrolidine-1-carboxamide
1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
(3aR,6aR)-2-methanesulfonyl-N-(3-phenylpropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[2-(4-fluorophenoxy)ethyl]-1,3-diazinane-2,4-dione
(1R,5R)-6-[(3,4-dimethoxypyridin-2-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
2-[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-(6-ethyl-4-methylquinolin-2-yl)-3-(hydroxymethyl)piperidin-3-ol
4-(3-methylbutyl)-3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
5-methanesulfonyl-2-methyl-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-4-amine
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-(benzyloxy)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-[(4-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
2-[(1-benzylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
2-{4-[2-amino-3-cyano-6-(4-hydroxyphenyl)-5-methylpyridin-4-yl]phenoxy}acetamide
1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
N-({7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
1-[5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
N-(5-chloro-2-methoxyphenyl)-3-(3-chlorobenzoyl)piperidine-1-carboxamide
(1R,5R)-6-{[4-(2-methylpropyl)phenyl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-2,4-dimethylpyrimidine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
1-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]urea
4-({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)piperazine-2-carboxylic acid
N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
5-methyl-5-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
5-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(2-hydroxyphenyl)acetamide
4-methyl-2-[4-(6-methylpyridazin-3-yl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
N-[(3S,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(thian-4-yl)piperazine
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-{1'-[(2S)-1-ethylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one