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4-{[1-(2-ethoxyacetyl)piperidin-3-yl]methyl}benzoic acid
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-methoxybenzamide
N-(piperidin-4-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(5-chloro-2-methoxybenzoyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-ethyl-4-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}pyrimidine
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
N-[(4-methoxyphenyl)methyl]-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(2,4-dimethoxyphenyl)ethan-1-one
2-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-methylquinoxaline
2-(1H-imidazol-1-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-(pyridin-2-ylmethyl)-3-(thiomorpholine-4-sulfonyl)benzamide
3-(2-ethylphenoxy)-1-(2-fluoro-4-methylbenzoyl)azetidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
5-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-2-(pyrrolidin-1-yl)benzonitrile
methyl 3-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
2-(benzyloxy)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
8-fluoro-4-oxo-N-[(4-sulfamoylphenyl)methyl]-1,4-dihydroquinoline-2-carboxamide
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(2-methylpropyl)acetamide
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][(2-methoxyphenyl)methyl](prop-2-en-1-yl)amine
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
2-hydroxy-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
4-(hydroxymethyl)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-ol
N'-(2,4-dimethoxyphenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanediamide
3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N,N-dimethyl-1-(thian-4-yl)piperidin-3-amine
2,2-difluoro-N-(2-{1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl}ethyl)acetamide
N-[5-(morpholin-4-yl)pentyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-butyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
methyl (3aS,6aS)-2-acetyl-5-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
4-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}-2-(trifluoromethyl)morpholine
2-(morpholin-4-yl)-3-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(6-methylpyridazin-3-yl)piperidin-3-ol
1-[4-({[2-(4-methyl-1H-imidazol-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
9-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[3-(pyridin-4-yl)propyl]acetamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(2-methylphenyl)piperidin-1-yl]butan-1-one
2-{[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]amino}pyridine-4-carbonitrile
1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyridin-3-yl)piperidin-4-ol
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-phenoxypropan-1-one
5-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1H-indole
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-methyl-1,3,4-oxadiazol-2-amine
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[2-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-fluorophenyl)acetamide