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N-(propan-2-yl)-1-[(1s,4s)-4-(2-methoxy-2-phenylacetamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(5-methoxyfuran-2-carbonyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
5-methyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}pyrimidin-2-amine
5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
[4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl 1-{[6-chloro-4-(4-methoxypiperidin-1-yl)quinazolin-2-yl]methyl}piperidine-2-carboxylate
1-(3-chlorophenyl)-4-(6-methoxyhexanoyl)-5-methylpiperazin-2-one
4-(4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)butan-1-ol
6-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
2-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)-6-methylpyridin-3-ol
ethyl 4-{[3-({1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine-1-carboxylate
[1-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)piperidin-2-yl]methanamine
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-[(2,3-dimethoxyphenyl)methyl]acetamide
3-methoxy-N-[(3S,5S)-1-methyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrrolidin-3-yl]propanamide
1-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
2-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
N-[4-(2-fluorophenoxy)phenyl]-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
(2S)-2-amino-3,3-dimethyl-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}butan-1-one
6-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,3-benzothiazole
1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidin-3-ol
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
3-methyl-N-(1-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopropanecarboxamide
5-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
(2S)-2-amino-3-(4-hydroxyphenyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
2-[1-cyclohexyl-4-(cyclopropylmethyl)piperazin-2-yl]ethan-1-ol
(2E)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
[1-(3-{[(adamantan-1-yl)amino]methyl}-7-fluoroquinolin-2-yl)piperidin-3-yl]methanol
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
N-(2,2-dimethylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methoxybenzamide
2-(3-methoxypropyl)-8-[2-(2,3,4-trifluorophenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(2S,4S)-N-ethyl-4-(2-hydroxyacetamido)-1-[(6-methylquinolin-5-yl)methyl]pyrrolidine-2-carboxamide
N-(1-{4-[(oxolan-2-ylmethyl)(propyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
N-cycloheptyl-4-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N-(4-butanamido-3-methoxyphenyl)quinoxaline-2-carboxamide
2-{1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-imidazol-2-yl}pyridine
2-(dimethylamino)-2-(4-fluorophenyl)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
(4aS,8aR)-6-(3-fluoropyridin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[5-(2-methoxyquinolin-3-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,3-diol
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]acetamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-(2-methylpropyl)pyridin-2-amine
3-(2-phenylethyl)-7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
7-(propan-2-yl)-2-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one