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1-[(4-fluorophenyl)methyl]-3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
1-(furan-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-{3-[3-(5-ethyl-2-methylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(methylamino)pyridine-4-carboxamide
N-(1-methoxybutan-2-yl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-methoxyethyl)-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-2-oxopentanamide
5-(methoxymethyl)-N-({7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylazepan-4-amine
N-[2-(1H-indol-3-yl)ethyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
3-methyl-1-(2-methylpropyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-2-[4-(4-{[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
5-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-benzothiazole
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
2-(furan-2-yl)-N-methyl-2-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
2-{1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}benzoic acid
6-(4-methoxy-3,5-dimethylphenyl)-N-methylpyridine-2-carboxamide
8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-[4-(4-fluorophenyl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(piperidine-1-carbonyl)piperidine
4-(4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
N3-[2-(3-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-{[3-(cyclohexylsulfanyl)propyl]carbamoyl}-1H-imidazole-4-carboxylic acid
2-methoxy-N-{[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
1-[1-(3-fluorobenzenesulfonyl)piperidin-3-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
2-(3-acetylphenyl)-2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}acetic acid
N-ethyl-3-(4-fluorophenyl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide
1-[4-phenyl-1-(2-propylpyridine-4-carbonyl)piperidin-4-yl]ethan-1-one
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methoxyphenyl)methyl]-N-methylacetamide
2-phenoxy-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-ethyl-3-[1-(1H-indole-5-carbonyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-methoxyphenyl)-4-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}piperazine
5-(3-methoxyphenoxymethyl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide
(1R,3S)-3-{4-[2-(3-methoxyphenoxy)ethyl]piperazine-1-carbonyl}cyclopentane-1-carboxylic acid
1-{5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carbonyl}piperidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
2-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(4-methylphenyl)piperazine-1-carboxamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]thiomorpholine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
(4aS,7aR)-1-(naphthalen-1-ylmethyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-methoxy-7-(4-methoxyphenyl)-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-1-(3-aminopropyl)-6-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
8-chloro-2-ethyl-4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine