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4-(1H-imidazol-1-yl)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
4-benzoyl-2-(2-phenylethyl)morpholine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(1,2-oxazol-3-ylmethyl)benzamide
2-{3-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]phenyl}ethan-1-amine
N-{3-[(4-methylphenyl)sulfanyl]propyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(2-methylpropanamido)methyl]benzoate
4-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,3-oxazole-5-carboxamide
3-[(2,4-dimethylphenyl)methyl]-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(2,5-dimethylphenoxy)-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
5-[3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1,3-oxazole
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
4-({1-[1-(1H-indol-5-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperazin-2-one
N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-2-[3-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
2-(cyclohex-1-en-1-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
6-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-({1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
(5-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}furan-2-yl)methanol
1-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
2-[(3,4-difluorophenyl)methyl]-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
dimethyl[(4-methyl-5-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
5-({3-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(ethylamino)pyrimidine-5-carboxamide
3-[4-(aminomethyl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
9-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[5-(2,5-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-1-methylpyrrolidin-2-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[2-(4-fluorophenyl)piperidin-1-yl]propan-1-one
2-methoxy-N-{2-methyl-1-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}acetamide
1-(2-methoxyethyl)-3-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
(1R,6S)-N-[2-chloro-5-(morpholin-4-yl)phenyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N4-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-[1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)-N-methylformamido]-N-methylbutanamide
8-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
methyl (2S,4S)-1-methyl-4-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}pyrrolidine-2-carboxylate
2-amino-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-4-carboxamide
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
methyl 3-{[(3-chlorophenyl)formamido]methyl}-5-(1,3-dimethyl-1H-pyrazole-5-amido)benzoate
ethyl 5-{[(oxolan-2-ylmethyl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(dimethylcarbamoyl)methyl]piperidine-2-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
ethyl 4-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidine-1-carboxylate
1-(butan-2-yl)-N3-[(2,4-difluorophenyl)methyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclobutyl-3-(naphthalene-1-carbonyl)piperidine
1-[7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
[1-(1-benzylpiperidin-4-yl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
3-(4-fluoro-3-methylphenyl)-6-propyl-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(2S)-1-acetyl-N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyrrolidine-2-carboxamide